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4-{[3-methyl-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl](pyridin-3-yl)methyl}morpholine
4-[2-(quinolin-8-yl)-1H-imidazol-1-yl]benzene-1-sulfonamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
2-{1-[1-(2-methyloxane-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
4-[7-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]morpholine
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanamide
3-[2-({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)ethyl]-1,3-oxazolidin-2-one
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
3-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)propanamide
1-{1'-[(2-fluoro-4-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
N-(1-{4-[2-(3,4-dimethylphenoxy)ethyl]phenyl}ethyl)acetamide
2-oxo-4-[2-(prop-2-yn-1-yloxy)phenyl]-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]acetamide
(1R,5R)-N,N-dimethyl-6-[4-(piperidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
2-methoxy-1-(4-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}piperidin-1-yl)ethan-1-one
3-tert-butyl-1-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}urea
N-[(2-methoxyphenyl)methyl]-2-[(pyridin-2-ylmethyl)amino]acetamide
1-[1-(2,3-dihydro-1-benzofuran-2-carbonyl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-{7,9-dioxo-8-azaspiro[4.5]decan-8-yl}-N-[(2-methoxyphenyl)methyl]acetamide
N-({4-hydroxy-1-[2-(methylsulfanyl)acetyl]azepan-4-yl}methyl)-2-phenoxyacetamide
1-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-4-phenoxypiperidine-4-carboxylic acid
N-[2-(2-hydroxyethoxy)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(2R,3R)-1'-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(dimethylamino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(5-methyl-1H-pyrazol-1-yl)propanamide
(3R,4R)-3,4-dimethyl-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidin-3-ol
2-{[ethyl(oxolan-2-ylmethyl)amino]methyl}benzonitrile
8-[(2,3-dimethyl-1H-indol-7-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylcyclohex-3-ene-1-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}(ethyl)amine
N-(3-methylbutyl)-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(5-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-[3-(1H-indazol-1-yl)propyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
5-methoxy-3-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1H-indazole
2-[2-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
2-benzyl-9-(1H-pyrazole-4-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
[(2-chlorophenyl)methyl][(5,6,7-trimethoxy-2-phenylquinolin-3-yl)methyl]amine
5-[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
2-[2-(dimethylamino)ethyl]-8-[2-(4-fluorophenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[3-(dimethylamino)phenyl]-4-methoxybenzamide
1-tert-butyl-4-({[6-(dimethylamino)pyrimidin-4-yl](methyl)amino}methyl)pyrrolidin-2-one
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methylpropanamide
(2R,3R,6R)-5-cyclopentanecarbonyl-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(1,5-dimethyl-1H-pyrazol-4-yl)-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetamide
N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
5-(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
N3-cyclooctyl-4-oxo-1-[2-(pyridin-2-yl)ethyl]-N5-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide