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8-{3-cyclopropyl-5-[(pyridin-4-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}quinoline
5-methanesulfonyl-2-methyl-N-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]pyrimidin-4-amine
(3aR,6aS)-5-[1-(4-fluorophenyl)piperidin-4-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2,4-dichlorophenoxy)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
2-({6-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-2-(trifluoromethyl)benzamide
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-cyclopentyl-4-fluoro-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}benzamide
2-[methyl(pyridin-4-ylmethyl)amino]-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
7-(3-chlorophenyl)-4-(3-methoxypropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1R,5R)-6-(2-methoxyethyl)-3-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
N-ethyl-3-(3-methoxyphenyl)-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
methyl({1-[1-(3-phenylbutyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)amine
2-[3-fluoro-5-(2-methylpropoxy)phenyl]-3-(piperidine-1-carbonyl)pyridine
1-{2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N-({3-methyl-7-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(piperidin-1-yl)acetamide
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-2,3,5,6-tetramethylbenzamide
methyl 6-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(4-chlorophenyl)-1-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-8-yl]butan-1-one
1-methyl-5-{4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazine-1-carbonyl}-1H-pyrrole-3-carbonitrile
1-(2-methyl-5-{1-oxa-8-azaspiro[4.5]decane-8-carbonyl}phenyl)imidazolidin-2-one
3-methyl-7-{2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-({4-[2-(furan-2-yl)pyrrolidine-1-carbonyl]furan-2-yl}methyl)morpholine
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-(piperidin-1-ylmethyl)benzamide
4-(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}azetidin-3-yl)morpholine
9-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-({4-[3-(morpholin-4-yl)propoxy]phenyl}methyl)piperazin-1-yl]ethan-1-one
4-{2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}-3-(4-fluorophenyl)piperazin-2-one
methyl 4-(2,6-diamino-3-cyano-5,6,7,8-tetrahydroquinolin-4-yl)thiophene-2-carboxylate
N-(1,2-oxazol-3-ylmethyl)-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
3-({[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}amino)propan-1-ol
[(3,4-dimethoxyphenyl)methyl](methyl)({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amine
3-(2,3-dimethylbenzoyl)-9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(3-methoxyphenyl)-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
4-(4-fluorophenoxy)-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidine-4-carboxylic acid
4-(pyridin-2-ylmethyl)-11-({[3-(trifluoromethyl)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(methoxymethyl)-5-methyl-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-4-(thiophen-2-yl)butanamide
1-{2-[3-fluoro-5-(propan-2-yloxy)phenyl]pyrimidin-4-yl}piperidin-4-ol
3-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
6-{2-[3-methyl-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]ethyl}-2,3-dihydropyridazin-3-one
2-(1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}azetidin-3-yl)pyridine
N-(3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-oxopropyl)methanesulfonamide
(1R,2R,4R)-N-[(2-propyl-1,3-thiazol-4-yl)methyl]bicyclo[2.2.1]hept-5-ene-2-carboxamide
3,3-dimethyl-1-({5-[(1-methyl-1H-indol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
1-[1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]-2-methylpropan-1-ol
3-(3-hydroxy-3-methylbutyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]benzamide
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]butanamide
7-(1,3-benzothiazol-2-yl)-4-[(3-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol