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4-(1-methyl-1H-pyrazol-4-yl)-N-(oxan-2-ylmethyl)pyrimidin-2-amine
1-methyl-1'-[4-(1H-pyrazol-1-yl)butanoyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-[4-(1-methoxypropan-2-yl)piperidin-1-yl]-5-methylpyrimidin-2-amine
2-(3-aminophenyl)-N-(propan-2-yl)pyridine-4-carboxamide
2-(5-acetylthiophen-3-yl)-1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
N-(2-{2-[4-(pyrimidin-2-yloxy)phenyl]-1H-imidazol-1-yl}ethyl)acetamide
1-(2-cyclohexylethyl)-3-hydroxy-3-{[methyl(prop-2-en-1-yl)amino]methyl}piperidin-2-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]pyridine-2-carboxamide
N-({1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
2-(1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-2-yl)pyridine
2,4-dimethyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1,3-thiazole-5-carboxamide
N-phenyl-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-amido}piperidine-1-carboxamide
ethyl 5-[(2-methyl-1H-indol-3-yl)methyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[1-(2-hydroxyphenyl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
7-[(4-fluorophenyl)methyl]-2-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
1-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
6-(quinolin-5-yl)pyridin-2-amine
3-{[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}-N-(furan-2-ylmethyl)propanamide
1-(1-methyl-1H-pyrrol-2-yl)-2-{4-methyl-3-oxo-1-oxa-4,9-diazaspiro[5.5]undecan-9-yl}ethane-1,2-dione
2-ethoxy-6-{[4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperazin-1-yl]methyl}phenol
N-(4-{[4-(3-methoxypyrazin-2-yl)piperazin-1-yl]methyl}phenyl)acetamide
1-{4-[2-(4-fluorophenyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-cyclohexyl-3-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}urea
2-{4-[(4,4-difluoropiperidin-1-yl)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
3-{[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
(1R,5S,6S)-3-[(4-methoxy-3-methylphenyl)methyl]-6-(4-methylpiperazine-1-carbonyl)-3-azabicyclo[3.1.0]hexane
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyacetyl)pyrrolidin-3-yl]-1-benzoxepine-4-carboxamide
1-benzyl-4-{[4-(2-propylpyrrolidine-1-carbonyl)-1,3-oxazol-2-yl]methyl}piperazine
(2R,3R,6R)-3-(4-fluorophenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
2-(methoxymethyl)-5-[(3-methyl-3-phenylpiperidin-1-yl)methyl]pyrimidine
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl][(2,4,5-trimethoxyphenyl)methyl]amine
3-(1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(5-methyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
11-methyl-4-[1-(pyridin-3-yl)propan-2-yl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-3-fluorobenzene-1-sulfonamide
1-methyl-4-{4-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine-1-carbonyl]phenyl}piperazine
N-{2-[3-(1H-indol-3-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
2-(3-hydroxyphenyl)-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
2-amino-4-(2-methoxyphenyl)-7-methyl-5H,7H-furo[3,4-b]pyridine-3-carbonitrile
N-[(2S,4R,6S)-2-benzyl-6-(2,5-dimethoxyphenyl)oxan-4-yl]acetamide
N-(1H-indazol-6-yl)-2-(3-methoxyphenyl)piperidine-1-carboxamide
7-chloro-4-[3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}pyrimidine-5-carboxamide
2-chloro-N,N-dimethyl-4-{[(2,2,2-trifluoroethyl)carbamoyl]amino}benzamide
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(piperidin-1-yl)ethan-1-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]pyrrolidin-3-yl]methanol