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(1S,5R)-3-(4-methyl-1H-imidazole-2-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(3R,4S)-3-(3-methyl-1H-pyrazole-5-amido)-4-propylpyrrolidin-1-yl]acetic acid
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1H-pyrazol-5-ylmethyl)amine
7-methyl-1-(pyridin-2-ylmethyl)-3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}-1,2-dihydroquinolin-2-one
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-(2,2-difluoroethyl)-4-(2-methoxyphenyl)piperazine
3-(3,4-dimethyl-1H-pyrazol-5-yl)-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]propanamide
3-(2-oxo-2-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}ethyl)-1,3-oxazolidin-2-one
N-(2,2-dimethyloxan-4-yl)-2-(4-hydroxypiperidin-1-yl)-6-(3-methylphenyl)pyridine-3-carboxamide
1-{2-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
1-(1-ethyl-1H-pyrazole-3-carbonyl)-2-[2-(thiophen-2-yl)ethyl]piperidine
7-cyclohexyl-2-(5-methylpyridin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(2-oxo-1,2-dihydropyridin-1-yl)propanamide
4-[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]-1-[(1R,2S)-2-propylcyclopropanecarbonyl]piperidine
N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1-benzothiophene-5-carboxamide
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)butan-1-one
1-[(1-propyl-1H-imidazol-2-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
5-({2-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,4-triazole
4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperazin-2-one
(3S,4S)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
4-methoxy-N-{[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]piperidine-4-carboxylate
2-(2-phenylethyl)-4-(pyridine-4-carbonyl)morpholine
1-[(3-fluorophenyl)methyl]-6-oxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-hydroxy-1-(pyridin-3-yl)ethyl]-1H-pyrazole-3-carboxamide
2-[2-(4-hydroxyphenyl)ethyl]-N-(pyridin-3-yl)piperidine-1-carboxamide
4-(2-ethyl-6-methylpyrimidin-4-yl)-1-[(3-methylphenyl)methyl]piperazin-2-one
ethyl 4-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}piperidine-1-carboxylate
2-(5-chloro-2-methoxybenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2,6-dimethoxypyridin-3-yl)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
1-[(5,6-dimethylpyrimidin-4-yl)amino]-3-(3-methoxyphenoxy)propan-2-ol
N-[1-(3-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]cyclobutanecarboxamide
N-(3-methoxyphenyl)-3-{[(3-methoxyphenyl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
N-[(8-methoxyquinolin-5-yl)methyl]-N,2-dimethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(3R,4S)-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(3-methoxyphenyl)pyrrolidin-3-amine
1-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-3-(furan-2-yl)propan-1-one
N-{4-[2-(2-cyclohexylpyrimidin-5-yl)-1H-imidazol-1-yl]-2-methoxyphenyl}acetamide
2-methyl-8-(6-phenylpyridazin-3-yl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-[3-(1H-indazol-1-yl)propyl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
1-(4-methylphenyl)-4-[3-(pyridin-4-yl)propanoyl]piperazin-2-one
6-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-2-carbonitrile
3-[(cyclopentylamino)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
7-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-(2-hydroxyethyl)-8-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
2-[2-(3-methyl-1H-pyrazol-1-yl)phenyl]acetic acid
N-(2H-1,3-benzodioxol-5-yl)-1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-amine
2-(4-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperazin-1-yl)-1,3-benzoxazole
4-(benzyloxy)-1-(3-phenyl-1,2-oxazole-4-carbonyl)piperidine
6-(2-fluoro-4-methoxyphenyl)-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(2R)-2-amino-N-ethyl-N-[(2-fluorophenyl)methyl]-4-methylpentanamide