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3-{2-[1-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]ethyl}phenol
4-methyl-6-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-5-(prop-2-en-1-yl)pyrimidin-2-amine
6-(cyclopropylmethoxy)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-4-(quinolin-2-ylmethyl)-1,4-diazepan-2-one
N-(4-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}phenyl)acetamide
3-cyclohexyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
7-(5-methylthiophen-2-yl)-4-(oxolan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(1H-indazole-3-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(2R,3R,6R)-5-(cyclopropanesulfonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N,N-dimethyl-2-(4-{2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetyl}piperazin-1-yl)acetamide
2-amino-1-[2-(5-{6-oxa-9-azaspiro[4.5]decane-9-carbonyl}thiophen-2-yl)pyrrolidin-1-yl]ethan-1-one
(1R,7S)-3-[4-(2-hydroxyethyl)phenyl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
6-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]pyridine-3-carbonitrile
1-({2-[butyl(methyl)carbamoyl]imidazo[1,2-a]pyridin-3-yl}methyl)piperidine-2-carboxamide
1-(1-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl)-N-(propan-2-yl)piperidine-4-carboxamide
methyl 3-[(3S,4R)-1-[(2E)-2-methylbut-2-en-1-yl]-4-(pyrrolidin-1-yl)piperidin-3-yl]propanoate
2-[1-(4-methoxyphenyl)piperidin-4-yl]-2,8-diazaspiro[4.5]decane
{4-fluoro-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
3-{[3-(diethylamino)pyrrolidin-1-yl]methyl}-6-methoxy-1,2-dihydroquinolin-2-one
N-[2-(7-{[5-(2-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxolane-2-carboxamide
2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-1-(piperidin-1-yl)ethan-1-one
N'-(2,5-dimethylphenyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]propanediamide
6-(2-methoxyphenyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyridazin-3-amine
4-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-(1-benzothiophen-2-ylmethyl)-5-[(3-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]methanol
2-(2-methoxy-5-methylphenyl)-5-(pyrrolidin-1-ylmethyl)pyridine
6-methoxy-3-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
(3S,7S)-5-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-triene-3-carboxylic acid
N-cyclopropyl-4-methoxy-2-({1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}oxy)benzamide
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-yl)ethan-1-ol
8-acetyl-2-(4-methylnaphthalene-1-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
7-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
5-(dimethylamino)-2-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydropyridazin-3-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-5-methyl-1,3-oxazole-4-carboxamide
1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
6-{2-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]ethyl}-2-methylpyrimidin-4-ol
8-[(3-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(2,2,2-trifluoroethyl)propanamide
4-[1-(2-phenylbenzoyl)piperidin-4-yl]pyridine
2-[2-(2-methylpropoxy)phenyl]-3-(piperidine-1-carbonyl)pyridine
N-(dicyclopropylmethyl)-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carboxamide
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N2-(2-methoxyethyl)-N4-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(3-methylbutan-2-yl)-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
N3-(1H-1,3-benzodiazol-2-ylmethyl)-N3-methyl-N5-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-butyl-1'-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-{[benzyl(methyl)amino]methyl}-N-[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
2-{[5-(1-ethyl-1H-pyrazol-3-yl)-4-(2-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid