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1-(5-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[3-(pyridin-2-yl)propyl]piperidin-4-amine
1-(azocan-1-yl)-2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-[(5-methylpyrazin-2-yl)methyl]-9-[2-(pyridin-3-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-1-(3-aminopropyl)-N-(cyclohexylmethyl)-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
1-{2-[5-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrrolidin-2-one
1-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1-methyl-3-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(6-methyl-2-propylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
4-({4-ethyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-N-methylbenzene-1-sulfonamide
2-[3-(1H-1,2,3-benzotriazol-1-yl)propanamido]-N,N-dimethylpropanamide
{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}[(1-ethyl-1H-pyrazol-4-yl)methyl]amine
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][1-(3-methoxyphenyl)propan-2-yl]amine
1-(4-methanesulfonylphenyl)-3-[1-(oxan-4-yl)piperidin-4-yl]urea
3-(2,3-dihydro-1H-inden-2-yl)-8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 4-oxo-4-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]butanoate
3-{3-[4-(pyrimidin-2-yl)piperazin-1-yl]propyl}-1H-indole
4-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}morpholine-2-carboxylic acid
4-[(3-{imidazo[1,2-b]pyridazin-3-yl}phenyl)methyl]morpholine
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
(1S,5R)-6-(1,3-thiazol-4-ylmethyl)-3-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]acetamide
5-ethyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-1,3-oxazole-4-carboxamide
N-[3-(4-chlorophenoxy)propyl]-4-(2,4-dioxoimidazolidin-1-yl)-N-methylbenzamide
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
ethyl 1-cyclobutyl-4-(3-phenylpropyl)piperidine-4-carboxylate
N4,5-dimethyl-N4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidine-2,4-diamine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(2-propoxybenzoyl)piperidine
2-[2-(dimethylamino)ethyl]-9-[(2-ethylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-acetyl-N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
methyl 1-(benzyloxy)-2-oxo-8-(thiolan-3-yl)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
1-({2-[1-(butan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}methyl)-1H-pyrazole
2-cyclopropyl-9-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(adamantan-1-yl)acetamido]-2-(4-fluorophenyl)acetic acid
3-{[(1-carbamoyl-1-methylethyl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-[1-(1H-indol-4-ylmethyl)piperidin-2-yl]propanoic acid
7-[(3,4-difluorophenyl)methyl]-2-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-methoxypyrazine
2-(2,5-dichlorophenyl)-3-methylpyrazine
7-(cyclobutylmethyl)-2-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
[(3S,4S)-4-(hydroxymethyl)-1-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}pyrrolidin-3-yl]methanol
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
5-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-N-propylpyrimidin-2-amine
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N,6-dimethyl-4-oxo-4H-pyran-2-carboxamide
N1,N1-dimethyl-N3-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidine-1,3-dicarboxamide
2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
2-{[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-3,5-dimethoxybenzoic acid
2-(2,4-dimethoxypyrimidin-5-yl)-N,N-bis(propan-2-yl)benzamide
3-ethyl-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N,4-dimethyl-1H-pyrazole-5-carboxamide