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N-[(3R,4S)-1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-propoxyacetamide
1-(carbamoylmethyl)-N-{2-[4-(dimethylamino)phenyl]ethyl}piperidine-4-carboxamide
3-[2-(dimethylamino)ethyl]-8-(3-hydroxypyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl N-(1-{4-[(4-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-1-oxopropan-2-yl)carbamate
2,6-dimethyl-4-({[1-(1-methyl-1H-pyrazol-5-yl)propyl]amino}methyl)phenyl acetate
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-ethyl-3,5-dimethyl-1H-pyrazole-4-carboxamide
(4S)-3,3,4-trimethyl-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-ol
N-cycloheptyl-3-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]propanamide
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methyl-5-{3-[3-(pyrrolidine-1-carbonyl)phenyl]phenyl}-1,3,4-thiadiazole
N-(4-methoxy-2-methylphenyl)-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]propanamide
4-ethyl-6-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]pyrimidine
(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-(pyrrolidine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
3-[2-(4-methoxyphenoxy)acetyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]benzamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-5-phenoxyfuran-2-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-(1,2-oxazol-3-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
2-(4-{[3-(pyridin-3-yl)azetidin-1-yl]sulfonyl}phenoxy)acetamide
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
3-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}pyridin-1-ium-1-olate
2-(3-methoxypropyl)-8-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
3-(2-{[4-(dimethylamino)-5-fluoropyrimidin-2-yl]amino}ethyl)-1,3-oxazolidin-2-one
N-[2-(4-benzylpiperazin-1-yl)ethyl]-4-ethyl-5-methylpyrimidin-2-amine
2-[2-({4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethyl]-5,6-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-[(2-chloro-3,4-dimethoxyphenyl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
8-[4,5-dimethyl-2-(1H-pyrrol-1-yl)thiophene-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
5-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-(pyridin-4-yl)pyrimidine
5-(3-methoxyphenyl)-4-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-2-(pyridin-4-yl)pyrimidine
5-ethyl-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-(2,5-dimethylphenyl)-3-[methyl(quinoxalin-2-ylmethyl)amino]propanamide
2-(3-methoxypropyl)-8-[(1-propyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{4-[3-(3-fluoro-4-phenylbenzoyl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-[(1S,2R)-2-[(1-ethylpiperidin-4-yl)amino]cyclobutyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N5-(butan-2-yl)-1-cyclopentyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclopropyl-5-[(4-hydroxyphenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{2-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}azepan-2-one
[(2,4-dimethoxy-3-methylphenyl)methyl](methyl)[1-(pyridin-3-yl)ethyl]amine
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-4-methylbenzamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3,4-dihydro-2H-1-benzopyran-6-carboxamide
2-tert-butyl-7,7-dimethyl-N-(oxan-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
4-(furan-2-ylmethyl)-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)piperazine-1-carboxamide
N-methyl-N-(prop-2-en-1-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
5-tert-butyl-3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-1H-pyrazole
N3-(2-methoxyethyl)-N3-[(3-methylthiophen-2-yl)methyl]piperidine-1,3-dicarboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-{[methyl(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(2-methoxyacetyl)pyrrolidin-3-yl]pyridine-3-carboxamide
4-(2,1,3-benzoxadiazol-4-ylmethyl)-1,4-oxazepan-6-ol
4-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-1,2,3-triazole
3-{5-[(1-phenyl-1H-pyrazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol