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(1R,5R)-6-[3-(3-methoxy-4-methylphenyl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(7-chloroquinolin-4-yl)azepan-3-amine
4-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidin-2-amine
2-{5-[2-(2-cyclohexyl-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridine
N-[2-(1H-indol-1-yl)ethyl]-N,2,6-trimethylquinoline-4-carboxamide
1-[(4aS,8aS)-4a-hydroxy-7-(5-methyl-1,3,4-thiadiazol-2-yl)-decahydro-2,7-naphthyridin-2-yl]-2-(dimethylamino)ethan-1-one
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-2,3-dimethyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-indole-7-carboxamide
ethyl 4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperazine-1-carboxylate
2-{[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}quinoline
5-(oxane-4-carbonyl)-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(4-{[1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
ethyl 4-(quinoxaline-5-amido)piperidine-1-carboxylate
(3aS,6aR)-5-(2-aminoacetyl)-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-(4,5-diphenyl-1H-imidazol-2-yl)-1-(propan-2-yl)pyrrolidin-2-one
[1-({1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
5-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
8-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N4-(pyridin-3-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-[2-(propylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
4,5-dimethyl-2-{2-[4-(pyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,3-benzodiazole
(3aR,6aR)-2-[(3-fluoro-2-methylphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2H-1,3-benzodioxol-5-yl)-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(dimethylamino)acetamide
N-[2-(N-methylmethanesulfonamido)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N3-[3-(2,5-dimethylphenoxy)propyl]-N3-methylpiperidine-1,3-dicarboxamide
4-[2-(4-fluorophenoxymethyl)-4-hydroxypyrimidine-5-carbonyl]-3-methylpiperazin-2-one
N-[1-(4-methanesulfonylphenyl)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-1H-pyrrole-2-carboxamide
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-2,7-dioxo-1,3-diazepane-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
4-ethyl-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[7-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
(7S,9aR)-6,9-dioxo-N-phenyl-7-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
2-[1-(2-propyl-1,3-thiazole-4-carbonyl)azetidin-3-yl]pyridine
N-methyl-3-(2-oxoazepan-1-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
2-[5-(1-benzylpiperidin-2-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-(naphthalene-2-carbonyl)-4-[2-(pyrrolidin-1-yl)ethyl]-1,4-diazepan-5-one
6-(benzyloxy)-4-(3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propanoyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
N-[1-(3,4-diethoxyphenyl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N,N-diethyl-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-sulfonamide
ethyl 1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[(2E)-3-phenylprop-2-en-1-yl]-8-[2-(pyridin-3-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
N-ethyl-5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxamide
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
2-chloro-4-[3-(piperidine-1-carbonyl)pyridin-2-yl]benzamide
N-[2-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-3-carboxamide
1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-2,4-dimethyl-1,4-diazepane
ethyl 4-(3-{[(2-methoxyphenyl)formamido]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)piperidine-1-carboxylate
4-{[2-chloro-5-methoxy-4-(propan-2-yloxy)phenyl]methyl}-1-methylpiperazine-2-carboxylic acid