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2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-(1H-pyrazol-5-ylmethyl)benzamide
(1S,5R)-6-[2-(4-chlorophenoxy)ethyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-(morpholin-2-yl)ethan-1-one
2-amino-3-ethyl-N-methyl-N-[3-(4-methylphenoxy)propyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
3-[(1-{[(pyridin-2-ylmethyl)carbamoyl]methyl}piperidin-4-yl)methyl]benzoic acid
methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})[1-(pyridin-2-yl)ethyl]amine
3-{[(1S,5R)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
2-(2-hydroxypropyl)-9-[3-(pyridin-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(4-fluorophenyl)phenyl]-7-methyl-2,7-diazaspiro[4.4]nonane-2-carboxamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(2,5-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2,2,2-trifluoroethyl)-1H-pyrazole-3-carboxamide
1-[7-(cyclobutylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-4-phenylbutane-1,4-dione
5-{[3-(4-cyclopentylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}isoquinoline
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]butanamide
[5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)furan-2-yl]methanol
methyl 2-[4-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)piperidin-1-yl]acetate
4-[(4-fluorophenyl)methyl]-1-(1-methylcyclopropanecarbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
3-acetamido-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)propanamide
5-tert-butyl-N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-1,3,4-oxadiazol-2-amine
(3S)-1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-ol
6-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
N-[1-benzyl-2-methyl-7-(thiomorpholine-4-carbonyl)-1H-1,3-benzodiazol-5-yl]-2-methylpropanamide
5-(2,6-difluorophenoxymethyl)-3-[3-(1H-pyrazol-1-yl)azetidine-1-carbonyl]-1,2-oxazole
methyl 4-[2-chloro-4-(cyclopentylcarbamoyl)phenoxy]piperidine-1-carboxylate
2,3-dimethyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}quinoxaline-6-carboxamide
N-benzyl-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{4-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
N-(4,6-dimethylpyridin-2-yl)-4-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)benzamide
(1S,5R)-3-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[(4-tert-butylphenyl)methyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
1-(oxane-2-carbonyl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
6-(azocane-1-carbonyl)-3-ethyl-3H-imidazo[4,5-b]pyridin-2-amine
1-cyclohexyl-3-(cyclopropylmethyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-({[(2-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)benzonitrile
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]acetamide
(3S,4S)-4-ethoxy-1-methyl-N-{2-methylpyrido[2,3-d]pyrimidin-4-yl}pyrrolidin-3-amine
7-methoxy-N,4-dimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]quinazolin-2-amine
8-[(3-chloro-2-fluorophenyl)methyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(3-chlorophenyl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
N-[(1R,2R)-2-(diethylamino)cyclohexyl]-N'-(2-methylphenyl)propanediamide
1-(4-methylpiperazin-1-yl)-3-[1-(thian-4-yl)piperidin-3-yl]propan-1-one
(3E)-2-{[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}-4-phenylbut-3-enoic acid
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]propanamide
5-fluoro-N4,N4-dimethyl-N2-[(1-propyl-1H-imidazol-2-yl)methyl]pyrimidine-2,4-diamine
N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}acetamide
2-{[4-(2,3-difluoro-4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-ethyl-1H-imidazole
3-[(2R,3R,6R)-5-{[2-(ethylamino)pyrimidin-5-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
3-(2-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
(2E)-N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]-3-(thiophen-2-yl)prop-2-enamide