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3-[1-(2-hydroxyethyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]-1-methyl-1,2-dihydroquinoxalin-2-one
2-methyl-5-{2-oxo-2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
4-(3-chloro-4-methoxyphenyl)-2,5-dimethylpyrimidine
(1S)-1-[1-(3-chloro-2-methylphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]propane-1,3-diamine
3-[4-methyl-3-(propan-2-yl)phenyl]-1-{3-[(pyridin-3-yl)amino]propyl}urea
8-(2-hydroxyacetyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{2-[4-(dimethylamino)phenyl]ethyl}-1-ethylpiperidine-2-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-(4-fluorophenoxy)azetidine
N,2-dimethyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,3-thiazole-4-carboxamide
N-[3-(1H-indol-1-yl)propyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
4-{[3-(3-fluorophenyl)phenyl]methyl}morpholine
1-(4-fluoro-2-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)-1H-pyrazole
(2R,3R)-3-[ethyl(methyl)amino]-1'-(1,3-thiazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-amino-N-[(2S)-oxolan-2-ylmethyl]-4-phenylpyrimidine-5-carboxamide
1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(methylamino)ethan-1-one
(3R,4R)-3,4-dimethyl-1-[1-(4-methylphenyl)cyclopropanecarbonyl]pyrrolidin-3-ol
4-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl}-2-{[4-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
5-tert-butyl-4-{[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]methyl}furan-2-carboxamide
N,5-dimethyl-1-propyl-N-[1-(pyridin-3-yl)propyl]-1H-pyrazole-4-carboxamide
4-(1-methyl-1H-pyrazol-4-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrimidin-2-amine
methyl N-(2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)carbamate
N-{3-methyl-4-[4-(2-oxopyrrolidin-1-yl)piperidine-1-carbonyl]phenyl}acetamide
5-(1-benzylpyrrolidin-3-yl)-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
4-[3-(3-chlorophenyl)-3-(2-hydroxyphenyl)propanoyl]-3,3-dimethylpiperazin-2-one
5-fluoro-N4,N4-dimethyl-N2-{2-[methyl(phenyl)amino]propyl}pyrimidine-2,4-diamine
4-[2-(naphthalen-1-yl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-(1,2,5-thiadiazole-3-carbonyl)piperidine
1-methyl-4-[4-(1,3-oxazol-5-yl)benzoyl]-1,4-diazepan-6-ol
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(3-fluorophenoxy)piperidin-1-yl]ethan-1-one
4-(1-aminocyclopropanecarbonyl)-7-(5-chloropyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,4R)-4-amino-1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperidine
2-[3-(dimethylamino)propyl]-9-(4-methylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-N-(4-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]carbamoyl}phenyl)furan-3-carboxamide
1-(adamantan-2-ylmethyl)-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
(2S,4R)-4-amino-1-{1-[(3,4-dimethylphenyl)amino]cyclohexanecarbonyl}-N-methylpyrrolidine-2-carboxamide
5-(2,3-dihydro-1-benzofuran-5-carbonyl)-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]quinoxaline-6-carboxamide
3-(2-methyl-1-benzofuran-5-yl)-1-(oxan-4-yl)urea
3,4,7-trimethyl-2-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-indole
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-3-methanesulfonylpropan-1-one
4-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-N,N-dimethyl-4-oxobutanamide
4-chloro-2-({4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)phenol
N-[2-methyl-4-(1H-pyrazol-3-yl)phenyl]pyridine-3-carboxamide
5-(4-acetyl-4-phenylpiperidine-1-carbonyl)-1-[2-(3-fluorophenyl)ethyl]piperidin-2-one
N-[1-(5-{[(4-methoxyphenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]cyclohexanecarboxamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-(oxan-2-ylmethyl)acetamide
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
4-[(3-methoxyphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
N-[2-(5-methylfuran-2-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide