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4-{1-[4-(5-fluoro-2-methoxyphenyl)phenyl]ethyl}morpholine
2-methyl-6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenol
4-cyclopentyl-N-{imidazo[1,2-a]pyridin-3-ylmethyl}pyrimidin-2-amine
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-(3-methylphenyl)ethan-1-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
4-{[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]methyl}benzonitrile
2-(adamantan-1-yl)-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}acetamide
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-cyclopropyl-15-methyl-13-oxo-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
2-(3-chloro-4-fluorophenyl)-2-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}acetic acid
N-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-N,2,2,6,6-pentamethylpiperidin-4-amine
2-cyclopropyl-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-methylpyrimidine-5-carboxamide
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-3-(1H-pyrazol-1-ylmethyl)benzamide
2-{[2-(furan-2-yl)pyrrolidin-1-yl]methyl}-4-hydroxyquinoline-6-carboxamide
6-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
{1-[1-(5-phenyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanamine
[(3,4-dimethoxyphenyl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
N-(1,3-benzothiazol-2-ylmethyl)-5-(2,6-difluorophenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
1-(diethylsulfamoyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
(4aS,7aR)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-fluorophenyl)-N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-3-oxopiperazine-1-carboxamide
(4aS,7aR)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-3-[3-(3-fluorophenyl)propanoyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,8aR)-1-(2-aminoethyl)-6-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-decahydro-1,6-naphthyridin-2-one
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
4-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-6-methylpyrimidin-2-amine
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-7-(thianthren-1-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(1-benzofuran-5-carbonyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
7-(cyclopropylmethyl)-2-(2-methylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(3S,4S)-4-({[3-(trifluoromethyl)pyridin-2-yl]amino}methyl)piperidin-3-ol
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amine
3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-N,N-dimethylaniline
2-[5-(oxane-2-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
(4aR,7aS)-1-(2-methoxyacetyl)-4-(1-methyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(hydroxymethyl)-N-(2,4,6-triethylphenyl)-1,4-oxazepane-4-carboxamide
3-(2-ethylbutyl)-8-(2-methoxypyridine-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4S,4aS,8aS)-4-phenyl-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}-decahydroquinolin-4-ol
N-[2-(3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)propyl]pyridine-4-carboxamide
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,5-dichlorophenyl)urea
2-({[(3R,4R)-1-[(3,5-dichlorophenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1-[(4-methylphenyl)methyl]pyrrolidin-2-one
3-(hydroxymethyl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-ol
1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-3-carboxamide
1-{5-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]thiophen-2-yl}ethan-1-one
N-[(3R,4S)-1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-4-propylpyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
6-{[(5-methyl-1,2-oxazol-3-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(3-methyl-1,2-oxazol-5-yl)acetamide
1-[(4aR,8aS)-1-[2-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
5-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2-(propan-2-yl)pyrimidine