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[(4-{[1-(2,3-dimethyl-1H-indole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
(3S,4S)-4-(propan-2-yl)-1-{[2-(propylamino)pyrimidin-5-yl]methyl}pyrrolidine-3-carboxylic acid
5-(1H-pyrazol-4-yl)quinoline
3-(2-propylpyrrolidine-1-carbonyl)-N-(pyrimidin-4-ylmethyl)benzene-1-sulfonamide
2-methyl-6-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-3-yl)-3,4-dihydropyrimidin-4-one
3-({methyl[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
(4aS,8aR)-6-(1H-pyrazole-3-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[2-(3-phenylpropyl)morpholin-4-yl]pent-4-en-1-one
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
N,2-dimethyl-4-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
1-cyclopropanecarbonyl-4-(2-phenylazetidine-1-carbonyl)piperidine
2-[4-(5-fluoro-2-methylphenyl)-2-methylphenoxy]acetamide
N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2,3-difluoro-6-methoxybenzamide
N-(2-{[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}ethyl)acetamide
3-(3-methoxypropyl)-1-(2-methylpyridin-4-yl)piperidine-3-carboxylic acid
[1-(4-fluorophenyl)ethyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
[1-methyl-4-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)piperazin-2-yl]methanol
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}pyrrolidin-3-yl]methanol
N3-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}piperidine-1,3-dicarboxamide
(benzylsulfamoyl)[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
(1S,3R)-3-amino-N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]cyclopentane-1-carboxamide
4-(2,3-dimethyl-1H-indole-7-carbonyl)-1,4-oxazepan-6-ol
8-[3-(dimethylamino)benzoyl]-2-(2-methylpropyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1H-imidazol-2-yl)benzamide
N,3,6-trimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1-benzofuran-2-carboxamide
(furan-2-ylmethyl)({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})(prop-2-yn-1-yl)amine
1-(cyclopropylmethyl)-4-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperazine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(5-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}furan-2-yl)benzonitrile
2-[({1-[(4-chloro-3-fluorophenyl)methyl]piperidin-4-yl}oxy)methyl]pyridine
1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3-(4-phenyl-1,2,3-thiadiazol-5-yl)urea
N-[(2R,4S,6S)-2-(3,5-difluorophenyl)-6-[1-(propan-2-yl)piperidin-4-yl]oxan-4-yl]acetamide
N-(3-methoxypropyl)-5-methyl-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
(1S,5R)-3-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
3-acetamido-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
(3R,4R)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
1-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
1-methyl-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H-indole-2-carboxamide
N-cyclopentyl-N-(3-phenylprop-2-yn-1-yl)-2-(1H-1,2,4-triazol-3-ylsulfanyl)acetamide
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
3-(4-methoxyphenyl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
2-ethyl-5-[4-(pyridin-3-yl)piperazine-1-carbonyl]pyrimidine
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(1H-imidazol-4-yl)ethyl]acetamide
N-[2-(2-fluorophenyl)ethyl]-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-(furan-2-ylmethyl)pyridin-2-amine
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(2-hydroxyphenyl)ethan-1-one
1-(4-{[2-(cyclopentyloxy)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one