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1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-hydroxypropan-1-one
2-methyl-1-[2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]-2-phenoxypropan-1-one
3-[(4-hydroxybutyl)sulfamoyl]-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
2-(4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
1-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)acetamide
1-cyclopentyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-N5-[phenyl(pyridin-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-{2-[(1R,2S,3R,4S)-3-amino-7-oxabicyclo[2.2.1]hept-5-ene-2-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
2-(2-{1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
(3S,4R)-3-benzyl-1-(1H-indole-5-carbonyl)-4-methylpiperidin-4-ol
4-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl[(5-propyl-1H-pyrazol-3-yl)methyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
5-chloro-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidin-2-amine
N-[1-(4-methoxyphenyl)-5-oxopyrrolidin-3-yl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
4-(2-methoxyethoxy)-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
(2S)-2-methoxy-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-2-phenylacetamide
3-ethyl-1-methyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
5-(1H-indole-6-carbonyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[2-(4,6-dihydroxypyrimidin-2-yl)ethyl]propanamide
3-[2-(3-fluorophenyl)ethyl]-1-(1,3-thiazol-2-ylmethyl)piperidine
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-ethoxyethan-1-one
1-(3,5-dimethoxyphenyl)-2-[(7-fluoroquinazolin-4-yl)amino]ethan-1-ol
2-oxo-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
(4aR,8aS)-1-(2-cyclohexylethyl)-6-[2-(thiophen-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-{[2-(difluoromethoxy)phenyl]methyl}-8-(pyrimidin-2-yl)-1,8-diazaspiro[4.5]decane
N-(2,4-dimethoxyphenyl)-3-[4-(4-methylphenoxy)piperidin-1-yl]-3-oxopropanamide
(2S,4S)-4-amino-N-ethyl-1-(5-methoxy-2,4-dimethylbenzenesulfonyl)pyrrolidine-2-carboxamide
2-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-methylazepane
1-[3-(3-ethylphenoxy)propyl]-1-methyl-3-(1-methyl-1H-pyrazol-4-yl)urea
3-[3-(3-methylthiophene-2-carbonyl)piperidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
[2-(4-fluorophenyl)ethyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
2-[1-(4-chlorophenyl)-5-oxo-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(oxolan-2-ylmethyl)acetamide
{4-[(4-chlorophenyl)methyl]-1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-4-yl}methanol
(1S,5R)-3-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[6-(diethylamino)pyridin-3-yl]-5-oxopyrrolidine-3-carboxylic acid
5-[2-(1H-1,3-benzodiazol-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[(3-methylthiophen-2-yl)methyl]-1,2-oxazole-3-carboxamide
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1-(propan-2-yl)-1H-imidazole
N-(2,3-dihydro-1H-inden-2-yl)-2-(3-fluoro-4-hydroxyphenyl)acetamide
1-[1-(5-methylthiophene-3-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(pentan-3-yl)acetamide
3-(3-hydroxyquinoxalin-2-yl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}propanamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[2-(methylsulfanyl)benzoyl]-decahydro-2,7-naphthyridine-2-carboxamide
2-[(4-fluorophenyl)methyl]-4-[(5-methylthiophen-2-yl)sulfonyl]morpholine
methyl 2-(1-{2-methylthieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl)acetate
N-cyclopentyl-1-ethyl-N-[(2-methoxyphenyl)methyl]-1H-pyrazole-3-carboxamide
2-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-4H-chromen-4-one
N-(1-ethyl-1H-pyrazol-5-yl)-2-{4-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-1H-pyrazol-1-yl}acetamide