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N-[2-(4-fluorophenyl)ethyl]-5-methyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
1-methyl-3-({4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazin-1-yl}methyl)-1,2-dihydroquinolin-2-one
6-methyl-2-{3-oxo-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carbonitrile
N-[(2,6-difluoro-3-methoxyphenyl)methyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-benzyl-N3-[2-(1H-indol-3-yl)ethyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(4-ethyl-3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
3-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}-1-methyl-1,2-dihydroquinolin-2-one
(3S)-4-(2-benzyl-1,3-thiazole-4-carbonyl)-3-ethylmorpholine
4-{3-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}-1H-pyrazole
4-methoxy-6-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
[(3-chlorophenyl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
3-{2-[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidine
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(4-fluorobenzoyl)piperidin-3-yl]piperazine
(1S,5R)-3-(2-phenoxyacetyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-4-({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}sulfamoyl)benzamide
3-(4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazol-1-yl)-1λ6-thiolane-1,1-dione
2-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2,8-diazaspiro[4.5]decane
2-(1,4-dimethyl-1H-indole-2-carbonyl)-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
1-{4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-2-methoxybenzoic acid
3-(1,3-benzothiazol-2-yl)-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}propan-1-one
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
5-[4-phenyl-1-(2-phenylpropyl)-1H-imidazol-5-yl]pyrimidin-2-amine
1-ethyl-N-[(1-ethyl-1H-indazol-3-yl)methyl]-3-methylpiperidine-3-carboxamide
2-methoxy-N,N-dimethyl-5-[({2-[(3-methylpyridin-4-yl)amino]ethyl}carbamoyl)amino]benzamide
1-(2-ethoxyphenyl)-4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
(1R,3s,6r,8S)-4-[2-(morpholine-4-carbonyl)pyridin-4-yl]-4-azatricyclo[4.3.1.13,8]undecane
5-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-3-yl}-N-[(4-methoxyphenyl)methyl]-4-methyl-1,3-thiazol-2-amine
2-methoxy-N-[4-methyl-3-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]carbamoyl}amino)phenyl]acetamide
1-[1-(2,2-difluoroethyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
2-methyl-5-{4-[1-(pyridin-2-yl)piperidine-3-carbonyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
2-(dimethylamino)-8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]methyl}-3-methoxyphenol
1-(2-methoxyphenyl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1H-pyrazole-4-carboxamide
3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine
5-methyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1H-1,3-benzodiazole-2-carboxamide
N-(cyclohex-1-en-1-ylmethyl)-7-(furan-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(5-phenyl-1,3,4-thiadiazol-2-yl)-N-[1-(pyridin-3-yl)propyl]piperidin-4-amine
2-(2-chloro-6-fluoro-3-methylbenzoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2,2-dimethyl-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxane-4-carboxamide
[5-(1,3-benzothiazol-2-yl)-2-fluorophenyl]methanol
3-{1-[1-(4-methoxyphenyl)propan-2-yl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
(1R,9aR)-1-{[4-(pyridin-4-ylmethyl)piperazin-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
4-[(2,5-dimethylphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1R,5R)-6-(1H-indole-2-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4,6-dimethyl-2-oxo-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide