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4-{[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]methyl}-1H-pyrazole-3-carboxylic acid
1-(2,3-dimethylphenyl)-N-[(2-fluoro-5-methoxyphenyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-(3-methyl-1H-pyrazol-1-yl)-1-{9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}propan-1-one
2-{4-[(3,5-dichloropyridin-4-yl)methyl]-1-(furan-2-ylmethyl)piperazin-2-yl}ethan-1-ol
3-{1-[2-(5-fluoro-2-methoxyphenyl)-1H-imidazol-1-yl]ethyl}-4-(2-methoxyethyl)-4H-1,2,4-triazole
1-{2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}imidazolidine-2,4-dione
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-3-ylmethyl)pyridin-2-amine
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-(dimethylamino)-2-(3-methylphenyl)acetamide
1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-(4-hydroxyphenyl)ethan-1-one
3-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridin-2-amine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-3-(1H-pyrazol-1-yl)benzamide
N,N-diethyl-6-methyl-2-(4-methylphenoxymethyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(4aS,8aR)-1-(3-aminopropyl)-6-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}quinoxaline-5-carboxamide
2-(2-hydroxypropyl)-9-[(1-propyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
7-[(pentafluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
2-(5-{[(1-methyl-1H-imidazol-2-yl)sulfanyl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
3,3,3-trifluoro-1-{3-[3-(morpholin-4-yl)-3-oxopropyl]piperidin-1-yl}propan-1-one
N-ethyl-2-(4-phenylpiperazin-1-yl)pyridine-3-carboxamide
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-(1-phenylcyclopropanecarbonyl)piperidin-3-yl]methanol
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-methylpiperidine-4-carbonitrile
ethyl 3-{[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]amino}propanoate
1-(dimethylsulfamoyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-[2-(hydroxymethyl)pyridin-4-yl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(2,3,6-trifluorobenzoyl)pyrrolidin-3-yl]methanol
N,1-diethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-5-methyl-1H-pyrazole-4-carboxamide
1-ethyl-6-methyl-3-[3-(pyridin-4-yl)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
N-[2-(diethylamino)ethyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-[3-chloro-4-(ethylcarbamoyl)phenyl]-3-(3-methylphenoxy)azetidine-1-carboxamide
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-[1-(2,6,8-trimethylquinoline-4-carbonyl)-1,4-diazepan-6-yl]acetic acid
2-(3-methoxypropyl)-9-[3-(pyridin-4-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)amine
2-propyl-N-[2-(pyridin-3-yl)ethyl]-1,3-thiazole-4-carboxamide
1-tert-butyl-5-(2-ethyl-4-methyl-1,3-oxazol-5-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1-(morpholin-4-yl)ethan-1-one
(3S)-N-tert-butyl-2-{[(pyridin-2-ylmethyl)carbamoyl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
methyl 3-{6-[(3-methoxyphenyl)methoxy]-4-[3-(methylsulfanyl)propanoyl]-2-oxo-1,4-diazepan-1-yl}propanoate
6-[2-(trifluoromethoxy)phenyl]-3H-imidazo[4,5-b]pyridine
4-{1-[4-(3-methoxyphenyl)phenyl]piperidin-4-yl}-1,4-oxazepane
N,N-dimethyl-1-[(2,7,8-trimethylquinolin-4-yl)methyl]pyrrolidin-3-amine
6-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
{1-[({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]cyclopropyl}methanol
2-{2-[2-(2-phenyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol