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4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-hydroxy-4-(methylsulfanyl)butan-1-one
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-(3-ethoxypropyl)-2,3-dihydro-1H-indene-2-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-3-phenyl-5-(thiomorpholine-4-sulfonyl)benzamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-(oxane-4-carbonyl)-4-(pyridin-4-yl)piperazine
3-({[5-(4-ethoxyphenyl)furan-2-yl]methyl}(methyl)amino)-N-methylbutanamide
5-fluoro-2-{1-[5-(5-methylfuran-2-yl)-1,2,4-triazin-3-yl]piperidin-4-yl}-1H-1,3-benzodiazole
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-3-phenyl-1H-pyrazole-4-carboxamide
8-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1,4-oxazepan-6-ol
8-methoxy-3-(piperidin-3-yl)-3,4-dihydroquinazolin-4-one
4-{[5-(1-cyclopentanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
(2S)-1-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]pyrrolidine-2-carboxamide
5-({3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1,3-dimethylimidazolidine-2,4-dione
N,N-dimethyl-5-{[4-(4-methylphenoxy)piperidin-1-yl]methyl}pyridin-2-amine
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
N-cyclopropyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
6-[1-(4-chlorophenyl)-3-hydroxypropan-2-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(ethylamino)-N-[1-(thiophen-2-yl)butyl]pyrimidine-5-carboxamide
8-fluoro-3-[2-(1-methylpiperidin-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-(2-ethyl-4-methyl-1,3-thiazol-5-yl)-1H-1,2,4-triazol-3-yl]acetamide
N'-(2,4-dimethoxyphenyl)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]propanediamide
1-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}naphthalen-2-ol
1-(4-chlorophenyl)-N-({1-[2-(pyrrolidin-1-yl)acetyl]piperidin-3-yl}methyl)cyclopropane-1-carboxamide
7-chloro-3-methyl-2-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}-1H-indole
4-ethyl-3-[1-(2-{imidazo[1,2-a]pyridin-3-yl}acetyl)piperidin-3-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-2-methylphenol
1-(3-{2-[2-(propan-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}propyl)-1H-indazole
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
5-[4-(5-ethylthiophene-2-carbonyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
5-cyclopropanecarbonyl-1'-(1-methylazepane-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-benzyl-3-ethyl-1-(2-ethylbenzoyl)-1,4-diazepan-5-one
2-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
3-(2-methoxypyridine-4-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
7-(cyclopropylmethyl)-2-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(benzylsulfanyl)-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyrimidine
5-(2,3-difluorobenzoyl)-2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-3-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1-ethyl-1H-pyrazole-3-carboxamide
2-[1-(2H-1,3-benzodioxol-5-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-N-(2-methylphenyl)acetamide
(3aS,6aS)-2-(2-hydroxyethyl)-5-{[3-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-1-[4-(3-chlorophenyl)piperazin-1-yl]ethan-1-one
7-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[3-(dimethylamino)propyl]-8-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-N-(2-methoxyethyl)-N-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-{[(3-propyl-1,2-oxazol-5-yl)methyl]amino}-N-(1,3-thiazol-2-yl)propanamide
N3-ethyl-N5-[(2-methoxyphenyl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl[(3-methylquinoxalin-2-yl)methyl](1,2-oxazol-3-ylmethyl)amine
dimethyl({[(1R,5S,6S)-3-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine