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N-(3-benzyl-1H-1,2,4-triazol-5-yl)-4-(4,6-dimethylpyrimidin-2-yl)piperazine-1-carboxamide
3-[2-({1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidin-4-yl}amino)ethyl]-1,3-oxazolidin-2-one
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}but-3-en-1-one
N-(cyclohexylmethyl)-3-(3-methoxypyrrolidine-1-carbonyl)benzene-1-sulfonamide
(1S,5R)-6-(2-methoxyethyl)-3-(5-methylpyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-[methyl({[4-(2-methylphenyl)phenyl]methyl})amino]ethyl}-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
8-(2,1,3-benzoxadiazol-4-ylmethyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-[(2R,3R)-2-ethoxy-1'-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
9-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-{[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-[(dimethylamino)methyl]-1-{[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-3-ol
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
7-[(3-fluoro-4-hydroxy-5-methoxyphenyl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}-2-methoxyphenol
1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-({[3-(thiophen-3-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)pyrimidine
1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methoxybenzoyl)piperazine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-3-azaspiro[5.5]undecan-9-amine
3-acetamido-N-[(4-methoxynaphthalen-1-yl)methyl]-N-(propan-2-yl)propanamide
(2S,4S)-N,N-diethyl-4-(4-hydroxybenzamido)-1-(2-methoxyacetyl)pyrrolidine-2-carboxamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-4-(pyridin-4-yl)pyrimidin-2-amine
1-[1'-(3-ethyl-1,2-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-[3-(1H-imidazol-1-yl)propyl]-3-{[(2-methoxyphenyl)methyl]amino}-5-(pyrrolidine-1-sulfonyl)benzamide
2-(2-{[methyl({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})amino]methyl}phenyl)-3,4,5,6,7,8-hexahydroquinazolin-4-one
5-butyl-1-(3-methylphenyl)-4-[2-(pyridin-4-yl)acetyl]piperazin-2-one
5-({3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
(3aR,6aS)-5-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(4-methylphenoxy)-1-{4-[2-(pyridin-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
2-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]pyrazine
1-(2-methoxyethyl)-4-({[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)pyrrolidin-2-one
N-(1-benzyl-5-oxopyrrolidin-3-yl)-2-(ethylamino)pyrimidine-5-carboxamide
4-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]phenol
1-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
N-methyl-4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-{1-[4-(trifluoromethyl)phenyl]pent-1-yn-3-yl}piperazine-1-sulfonamide
N-methyl-4-(4-methylphenoxy)-N-[1-(1,2-oxazol-3-yl)ethyl]piperidine-4-carboxamide
3-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-3-yl)propanamide
2-{2-[(3S)-3-ethylmorpholin-4-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(3-phenylpropyl)-N-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
(1R,5S,6S)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}[4-(methylsulfanyl)butan-2-yl]amine
3-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]quinoline
6-(2-fluoro-5-methoxyphenyl)-N,N-dimethylpyridine-2-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(pent-4-enoyl)piperidin-4-yl]oxy}benzamide
5-(4-benzylpiperidine-1-carbonyl)-N-phenylpyrimidin-2-amine
2-methoxy-1-{3-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]piperidin-1-yl}ethan-1-one
[2-(2,5-dimethylphenoxy)ethyl](methyl)[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine