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1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-(furan-2-carbonyl)-1,4-diazepan-6-ol
2-{[4-(4-benzyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenol
methyl 8-(1H-indol-3-ylmethyl)-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-{2-[(4-fluoropiperidin-1-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}pyridin-2-ol
N,1-dimethyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
2-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-3-methylquinoline
1-[2-(morpholin-4-yl)phenyl]-5-oxopyrrolidine-3-carboxylic acid
4-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methylphenol
1-methyl-4-[4-(1H-pyrazol-4-yl)butanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
[1-(1-benzothiophen-2-ylmethyl)-4-(oxan-2-ylmethyl)piperidin-4-yl]methanol
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]azepan-3-amine
4-(3-ethyl-1H-indole-2-carbonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{[tert-butyl(3-phenylprop-2-yn-1-yl)amino]methyl}pyridine-3-carboxylic acid
5-{[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}-1-[(2-methylphenyl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethan-1-one
4-methyl-N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pentanamide
5-({4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)-2-methoxyphenol
methyl 5-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-(morpholin-3-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]ethan-1-one
(4aS,7aR)-1-[3-(methylsulfanyl)propanoyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-(4-methyl-1,3-thiazole-5-carbonyl)-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
5-(3-methylfuran-2-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-methyl-3-phenyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,2-oxazole-5-carboxamide
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-(3-phenylpropyl)piperidine
1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)-4-methylpiperidine
2-{[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzonitrile
2,5,7-trimethyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-1-(5-methyl-1,3,4-thiadiazol-2-yl)urea
2-{1-[(2-methylphenyl)methyl]-4-(1,3-thiazol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N,1,6-trimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(propan-2-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1,2-oxazole-3-carboxamide
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-{[(3R,4R)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}-2,5,7-trimethylquinoline-4-carboxamide
1-(4-{1,9-dioxaspiro[5.5]undecan-4-yl}piperazin-1-yl)-2-phenoxyethan-1-one
5-chloro-2-(4-{[3-(prop-2-en-1-yloxy)phenyl]methyl}piperazin-1-yl)pyrimidine
1-[2-(3-chlorophenyl)ethyl]-4-[(6-ethylpyrimidin-4-yl)amino]pyrrolidin-2-one
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carboxamide
2,6-dimethoxy-4-({[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amino}methyl)phenol
4-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)-1λ6-thiomorpholine-1,1-dione
1-{4-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-4-oxobutyl}piperidin-2-one
6-{4-[2,5-dioxo-4-(pyridin-3-yl)imidazolidin-4-yl]piperidin-1-yl}pyridine-3-carboxamide
4-{3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-1,4-oxazepane
1-(2-phenylethyl)-4-(4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}phenoxy)piperidine
1-(2-{[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]amino}pyrimidin-4-yl)piperidin-4-ol
methyl[2-(morpholin-4-yl)propyl]{[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}amine
1-(2-methoxy-5-{[methyl(2-phenylethyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
6-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one