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N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2,5-dimethylpyrimidin-4-amine
(3aS,6aS)-2-cyclohexyl-5-{[methyl(phenyl)carbamoyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-butyl-8-(1-methyl-1H-indole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
6-[(diethylamino)methyl]-N-[(1-ethyl-1H-imidazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}-1,2-oxazole-3-carboxamide
[(2S,6S)-4-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[(5-phenylthiophen-2-yl)methyl]-decahydro-2,7-naphthyridine-2-carboxamide
1-(1-benzyl-5-oxopyrrolidin-3-yl)-3-(1-cyclohexyl-1H-pyrazol-5-yl)urea
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
(3aS,6aS)-2-(1-benzoylpiperidin-4-yl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-4-(2-oxopyrrolidin-1-yl)benzamide
3-[1-(1-methyl-1H-1,3-benzodiazol-5-yl)-N-(2-phenylethyl)formamido]propanamide
methyl 6-[(2,4-dimethylphenyl)methyl]-2-[(propan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-[1-cyclohexyl-5-(oxolan-3-yl)-1H-1,2,4-triazol-3-yl]benzamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(furan-2-amido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-[(3,3-dimethylcyclohexyl)amino]-3-(3-methoxyphenoxy)propan-2-ol
N,1-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-3-propyl-1H-pyrazole-5-carboxamide
7-fluoro-4-(1,4-oxazepane-4-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
(2S)-2-{[5-(4-methylphenyl)-1H-pyrazol-3-yl]formamido}-3-phenylpropanamide
4-[5-(2-methylbenzamido)-1H-pyrazol-1-yl]-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
1-{2,4,6-trimethyl-3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]phenyl}ethan-1-one
3-[2-(4-fluorophenyl)ethyl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine
2-ethyl-4-{1-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methanesulfonamido-N-methylpropanamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5,7-dimethyl-2,1,3-benzoxadiazole-4-sulfonamide
2-(2-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amino]methyl}phenoxy)ethan-1-ol
(3S,4R)-1-(3-ethoxypropanoyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-{2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[(2-butyl-1H-imidazol-4-yl)methyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(3,4-dichlorophenyl)-4-(2-methoxy-4-methylbenzoyl)morpholine
N-(oxan-4-ylmethyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
8-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-2-(2-methylpropyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[(4-chlorophenyl)methyl]-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-6-oxopiperidine-3-carboxamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-3-sulfamoylthiophene-2-carboxamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]propan-1-one
4,6-dimethyl-2-oxo-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-methyl-N-[(3-methyloxetan-3-yl)methyl]-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
2-hydroxy-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyridine-3-carboxamide
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
2-{[methyl({7H-pyrrolo[2,3-d]pyrimidin-4-yl})amino]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[(6-methylpyridin-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
N-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-3-propoxypiperidine-1-carboxamide
4-(hydroxymethyl)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}azepan-4-ol
4-(4-chloro-2-methylbenzoyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-amino-3-ethyl-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-phenyl-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
1-methyl-4-(3-methylbut-2-enoyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-ethyl-6-(4-fluorophenyl)-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine