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4-(dimethoxy-1,3,5-triazin-2-yl)phenol
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
6-(4-chloro-2-methoxybenzoyl)-2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-(2-phenylpropyl)-8-[3-(pyridin-3-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(2-methoxyethoxy)-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine
3-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-6-ethyl-3,4-dihydroquinazolin-4-one
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(2-hydroxyethoxy)ethyl]acetamide
4-(2-chloro-4-methoxyphenoxy)-1-methylpiperidine-4-carboxylic acid
4-[4-(dimethylamino)benzoyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-(3-fluorophenoxymethyl)-N-(quinolin-3-ylmethyl)-1,3-oxazole-4-carboxamide
5-(4-methoxyphenyl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}furan-2-carboxamide
2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyridine-3-carboxylic acid
4-methoxy-N-methyl-3-[2-(morpholin-4-ylmethyl)phenyl]benzamide
1-phenyl-4-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperazine
2-chloro-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-(1H-pyrazol-1-yl)benzamide
1-(2-phenylethyl)-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(4-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[(2-methoxypyrimidin-5-yl)methyl]-2-methyl-1,4-diazepan-5-one
5-[3-(morpholin-4-ylmethyl)phenyl]-2,3-dihydro-1H-indol-2-one
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-3-(1H-1,2,4-triazol-1-yl)propanamide
1-{9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-phenylethan-1-one
2-(3-methoxyphenyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,3-benzoxazole-6-carboxamide
5-{5-[(S)-methoxy(phenyl)methyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1,3-dimethyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-(2-methanesulfonylethyl)-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-[(1-ethyl-1H-indol-3-yl)sulfanyl]-N-(1,2-oxazol-3-ylmethyl)acetamide
3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-N-{[4-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-4-yl}methanesulfonamide
4-[3-(2,5-dimethylfuran-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methyl-6-(1H-pyrazol-1-yl)pyrimidine
3-(dimethyl-1,2-oxazole-4-carbonyl)-9-(3,3-dimethylbutyl)-3,9-diazaspiro[5.5]undecane
2-[(3,5-difluorophenyl)methyl]-8-(2-hydroxyethyl)-2,8-diazaspiro[4.5]decan-3-one
(3R,4R)-4-methyl-1-{4-[(4-methylpiperazin-1-yl)methyl]benzoyl}-3-(propan-2-yl)pyrrolidin-3-ol
N-(2-methoxyethyl)-2-phenoxy-N-(thiophen-3-ylmethyl)acetamide
4-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-2-yl)methyl]morpholine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,7-dimethylquinoline-4-carboxamide
2,8-dimethyl-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]quinoline-4-carboxamide
1-(cyclopropylmethyl)-N-ethyl-5-(1H-indole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1-(pyridin-2-yl)piperidine-3-carboxamide
(1R,3S)-N3-ethyl-1,2,2-trimethyl-N1-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]cyclopentane-1,3-dicarboxamide
7-(3-chlorophenyl)-4-(1,3-thiazol-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
1-[4-({[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}amino)piperidin-1-yl]ethan-1-one
N,1-dimethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
1-(3-methylphenyl)-4-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}pyrrolidin-2-one
4-hydroxy-2-methyl-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]pyrimidine-5-carboxamide
N-methyl-N-[2-(oxan-2-yl)ethyl]-1H-1,2,4-triazole-5-carboxamide
1-(2-methyl-5-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
6-(3-fluoro-4-methoxyphenyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide