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N-{1-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-{4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl}-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
1-ethyl-N-(furan-2-ylmethyl)-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 2-({1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]piperidin-4-yl}formamido)acetate
5-(oxane-2-carbonyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(4-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
5-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
2-(3-methyl-4-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
1-[(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}thiophen-3-yl)methyl]piperidine
6-(2-aminoethyl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrimidin-4-amine
(3R,4R)-4-cyclobutyl-3-methyl-1-(1,3-thiazol-2-yl)piperidin-4-ol
N-(3-cyano-4-ethoxyphenyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carboxamide
1-[4-(1H-imidazol-4-ylmethyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-9-yl]-2-phenoxyethan-1-one
ethyl 2-[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]-1,3-oxazole-4-carboxylate
N-[(3S,4R)-4-(4-methylphenyl)-1-[(3-methylquinoxalin-2-yl)methyl]pyrrolidin-3-yl]acetamide
1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
N-[(4-fluorophenyl)methyl]-N-(1-hydroxybutan-2-yl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(4-fluoro-3-methoxyphenyl)methyl]-4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
4-methyl-2-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
2-(1H-1,3-benzodiazol-1-yl)-1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(2E)-3-phenylprop-2-en-1-yl]amino)ethan-1-ol
1-({2-[3-(piperidin-1-yl)propoxy]phenyl}methyl)pyrrolidin-3-amine
2-methyl-8-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[(2-ethylpyrimidin-5-yl)methyl]-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(3-methylpyridin-4-yl)methyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-3-carboxamide
6-[3-methyl-4-(propan-2-yl)piperazin-1-yl]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
8-(3-fluorobenzoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
[4-(2-phenoxyethyl)-1-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-yl]methanol
N-(cyclohex-1-en-1-ylmethyl)-3,4-dimethyl-5-sulfamoylbenzamide
N-{[5-(3-methoxypyrazin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
(2S,4S)-4-amino-N-methyl-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidine-2-carboxamide
2,2-dimethyl-N-[3-(4-methylbenzenesulfonamido)propyl]oxane-4-carboxamide
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[(2-oxo-1,2-dihydropyridin-1-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
N'1-[(3R,4S)-1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
4-(4-chlorophenyl)-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methylbutanamide
9-[2-(2-ethoxyethoxy)benzoyl]-3,9-diazaspiro[5.6]dodecane
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(2-methylpropanoyl)piperidin-3-yl]propanamide
2-(2,3-dimethylphenoxy)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
4-(3-{[1-(2-chlorobenzoyl)piperidin-4-yl]oxy}benzoyl)morpholine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]pyridine-3-sulfonamide
[(3R,4R)-1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[(cyclopropylamino)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
(4aS,7aR)-1-[(3,5-dimethylphenyl)methyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(furan-2-yl)-2-oxoacetamide