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N-[2-(1H-imidazol-2-yl)ethyl]-5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-amine
1-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]urea
8-(2,3,5,6-tetramethylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
(1R,5R)-6-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
6-[1-(5-chlorothiophene-2-carbonyl)piperidin-4-yl]-2-methyl-3,4-dihydropyrimidin-4-one
(1R,5R)-6-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
2-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
1-methyl-1'-[2-(1H-pyrazol-1-ylmethyl)propanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-methyl-8-[(6-methyl-4-oxo-1,4-dihydroquinolin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(4H-1,2,4-triazol-4-yl)ethan-1-one
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl](methyl){[2-(methylsulfanyl)phenyl]methyl}amine
N-[(4-fluoro-3-methoxyphenyl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(4-chlorophenyl)-2-[4-(piperidin-1-yl)butanamido]acetic acid
9-(5-methylpyridine-2-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-1-(6-methoxypyrimidin-4-yl)pyrrolidine-3-carboxamide
2-{[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
4-({1-[1-(ethoxycarbonyl)piperidin-4-yl]pyrrolidin-3-yl}methyl)benzoic acid
8-(1-methoxypropan-2-yl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aS)-2-(ethanesulfonyl)-5-(2-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2,5-dimethyl-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
methyl 4-[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)carbamoyl]butanoate
5-methanesulfonyl-1'-(1-methyl-1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-methyl-2-{1-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
(3R)-1-[3-(azocane-1-carbonyl)benzenesulfonyl]pyrrolidin-3-ol
4,6-dimethyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]quinolin-2-amine
N-[(2S,4R,6R)-2-(4-chloro-1-methyl-1H-pyrazol-3-yl)-6-cyclohexyloxan-4-yl]acetamide
1-{[2-(cyclopentyloxy)phenyl]methyl}-4,4-difluoropiperidine
4-ethyl-1-methyl-3-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-hydroxy-3-{[methyl(oxan-4-yl)amino]methyl}-1-(2-phenylethyl)piperidin-2-one
6-ethyl-5-methyl-N4-{2-[(pyridin-3-yl)amino]ethyl}pyrimidine-2,4-diamine
2-(3-oxo-9-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-2-yl)acetamide
(butan-2-yl)(pyridin-3-ylmethyl){[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
2-{2-[3-(dimethylamino)pyrrolidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
[(3R,4R)-1-(3-methyl-1,2-oxazole-5-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-(furan-3-ylmethyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-(1-ethylpiperidin-4-yl)-1-[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
3-(4-hydroxybenzamido)-4-(2-methylpiperidin-1-yl)benzamide
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-propylpiperidine-1-carboxamide
N-[(2-chlorophenyl)methyl]-6-fluoro-N-(2-methoxyethyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-[({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)amino)methyl]-7-methoxy-1,2-dihydroquinolin-2-one
3-{2-[3-(3-ethylphenoxy)azetidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}pyridin-2-amine
1-(1-{1-[(2-methyl-1-benzothiophen-3-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
3,5-dimethoxy-2-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)benzoic acid
[3-methyl-1-oxo-1-(3-oxo-4-phenylpiperazin-1-yl)butan-2-yl]urea
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide