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3,5-dimethoxy-2-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)benzoic acid
3-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}-N-(1-methyl-1H-1,2,3-triazol-4-yl)benzamide
N-[(3S,4R)-1-(6-hydroxyhexyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
4-[(2-ethylpyrimidin-5-yl)methyl]-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
3-cyclopropaneamido-N,4-dimethyl-N-[(3-methylthiophen-2-yl)methyl]benzamide
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(propan-2-yl)pyridine-4-carboxamide
N-[2-(dimethylsulfamoyl)ethyl]-2-hydroxy-2-[4-(trifluoromethyl)phenyl]acetamide
4-{4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
methyl({[5-(oxolan-2-yl)thiophen-2-yl]methyl}){[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
1-(2-ethoxypyridine-3-carbonyl)-4-(2-methylphenyl)-1,4-diazepane
5-(3-acetylphenoxymethyl)-N-[1-(2-chlorophenyl)ethyl]-1,2-oxazole-3-carboxamide
9-(3-aminothiophene-2-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(pyrrolidin-1-yl)pyridine-3-carboxamide
N-[(2S,4R,6R)-2-(6-methoxypyridin-3-yl)-6-(propan-2-yl)oxan-4-yl]benzamide
N-[(4-fluorophenyl)methyl]-3-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
1-(2-methyl-5-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}phenyl)imidazolidin-2-one
1-{3-[7-(1-benzothiophen-3-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}imidazolidin-2-one
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2-propyl-1,3-thiazole-4-carboxamide
6-(4-aminopiperidin-1-yl)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]pyridine-3-carboxamide
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
2-(4-chloro-1H-pyrazol-1-yl)-1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]ethan-1-one
1-(5-fluoropentyl)-2-oxo-3-[2-(pyridin-2-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-(2-hydroxyethyl)-1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
[(3R,4R)-1-(3-fluoropyridin-4-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-2-methyl-3-[(pyridin-2-ylmethyl)amino]benzamide
1-methyl-2-phenyl-4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazine
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]acetamide
5-{1-[2-(dimethyl-1,3-thiazol-4-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-{9-[(3,5-dimethylphenyl)carbamoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
3-methyl-1-phenyl-4-{1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-5-amine
4,6-dimethyl-2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carbonitrile
2-methyl-6-[1-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-1,2,3-triazol-4-yl]pyridine
5-benzyl-1-(4-methylphenyl)-4-(2-methylpropanoyl)piperazin-2-one
(3aR,6aS)-5-(1-benzofuran-2-sulfonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3R,4S)-1-(carbamoylmethyl)-4-propylpyrrolidin-3-yl]-4-chloro-1,5-dimethyl-1H-pyrazole-3-carboxamide
9-(2-fluorobenzoyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-{[3-(methylsulfanyl)phenyl]methyl}-N-(propan-2-yl)-2-(thiophen-2-yl)acetamide
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
1-cyclopentyl-6-oxo-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperidine-3-carboxamide
2-[1-(2-fluorophenyl)-5-[2-(propan-2-yl)-1,3-thiazol-4-yl]-1H-1,2,4-triazol-3-yl]acetamide
1-cyclopentyl-N-[2-(1H-indol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
1-(3-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenyl)ethan-1-one
4-{[4-(isoquinolin-1-yl)piperazin-1-yl]methyl}benzoic acid
2-(3-methoxyphenoxy)-1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}ethan-1-one
3-(2-chlorophenyl)-N-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-3-phenylpropanamide
4-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
6-[4-(4-fluorophenyl)-4-oxobutanoyl]-N-[2-(3-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide