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1-(3,5-dimethylphenyl)-4-(3-ethyl-1H-pyrazole-4-carbonyl)piperazin-2-one
2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}benzene-1,3-diol
2-(2-fluoro-5-methoxyphenyl)-5-methyl-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
methyl 5-[(2,3-dihydroxypropyl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-({4-hydroxy-1-[(2-methyl-1,3-thiazol-4-yl)methyl]azepan-4-yl}methyl)thiophene-2-carboxamide
3-methyl-8-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[(1-{6-[(furan-3-ylmethyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
3-{[1-(5-phenyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-yl]methyl}benzamide
(1R,5S,6R,7S)-3-(2-aminoethyl)-6-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]decan-4-one
5-(2,5-dimethylfuran-3-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
methyl 5-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-1-methyl-1H-pyrazole-3-carboxylate
1-[(3-fluorophenyl)methyl]-4-{2-oxo-1-oxaspiro[4.4]nonane-4-carbonyl}piperazin-2-one
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(naphthalen-1-yl)ethan-1-one
4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(3-methoxyphenyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
2-(1-ethyl-1H-pyrazol-4-yl)-6-methoxy-N,N-bis(propan-2-yl)benzamide
(3S,4R)-1-(6-fluoro-4-methylquinolin-2-yl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
5-[5-(2-chlorophenyl)furan-2-yl]-3-methyl-1,2,4-oxadiazole
2-{5-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1H-pyrazol-3-yl}phenol
N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2,3-dihydro-1,4-benzodioxine-5-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
2-{[(3S,5S)-5-(ethylcarbamoyl)-1-[(5-methylfuran-2-yl)methyl]pyrrolidin-3-yl]amino}pyridine-3-carboxamide
2-[(cyclohexylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-{3-cyclopentyl-5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
4-{2-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}morpholine
6-methyl-4-[2-(prop-2-en-1-yloxy)phenyl]-5-(1,2,3,6-tetrahydropyridine-1-carbonyl)-1,2,3,4-tetrahydropyrimidin-2-one
5-methyl-2-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]pyrimidin-4-amine
2-[1-(5-chloropyridine-3-carbonyl)pyrrolidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
3-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
2-{methyl[(1-{[1-(2-methylpentyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]amino}ethan-1-ol
7-chloro-2-(furan-2-yl)-8-methyl-N-(1,2-oxazol-3-ylmethyl)quinoline-4-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-2-(1-methylcyclopropanecarbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
3-[(2H-1,3-benzodioxol-5-yl)amino]-N-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)piperidine-1-carboxamide
8-[(4-chloro-3-fluorophenyl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3,5-dichloro-4-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}pyridine
ethyl 1-{[1-(1H-1,3-benzodiazol-2-yl)-4-(ethoxycarbonyl)-1H-pyrazol-5-yl]methyl}piperidine-3-carboxylate
1-[3-(4-{2-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine-1-carbonyl)phenyl]imidazolidin-2-one
2-fluoro-N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)benzamide
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(thiophen-3-yl)acetamide
N-benzyl-1-[2-(3-methoxypropyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
6-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-9H-purin-2-amine
1-[1-(2-phenylethyl)-5-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
(3aR,6aS)-5-(2,1,3-benzoxadiazol-5-ylmethyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(5-methylthiophen-2-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(pyridin-2-ylmethyl)-9-(pyrimidin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(propan-2-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1,2-oxazole-5-carboxamide
2-ethyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-4-methyl-1,3-oxazole
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide