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2-(2-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}ethyl)pyridine
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
3-({4-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]piperidin-4-yl}oxy)-2-methylpyridine
3-(3-fluoro-4-methoxyphenyl)-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-(2-methylphenyl)-1H-pyrazole
N-({1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
2-(dimethyl-1,3-thiazole-5-carbonyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
2-cyclopropyl-1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-[5-(1H-imidazol-2-yl)pyrimidin-2-yl]benzenesulfonamide
(3S,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
(2R,3R)-3-(dimethylamino)-1'-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
methyl 4-[4-(5-fluoropyridin-2-yl)piperazin-1-yl]benzoate
N-{1-[4-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)phenyl]-1H-pyrazol-4-yl}oxane-4-carboxamide
2-{[(1S,5R)-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
2-(2-fluoro-4-methylphenyl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(3-methylphenyl)piperidine
1-{4-[(3-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-4-methoxyphenyl)methyl]piperazin-1-yl}ethan-1-one
3-ethoxy-1-(7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
7-(3-chlorophenyl)-4-[6-(1-hydroxyethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[4-(but-3-yn-1-yloxy)phenyl]methyl}-N-(oxolan-2-ylmethyl)cyclohexanecarboxamide
N-(2-methoxyethyl)-N-(naphthalen-1-ylmethyl)-1-phenyl-1H-1,2,3-triazole-4-carboxamide
1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-3-phenylpiperidine
1-[5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]azocane
1-(3-ethyl-1H-pyrazole-4-carbonyl)-4-(4-methoxyphenyl)-2-methylpiperazine
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
1-[(4-phenylphenyl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
2-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]-3-methylquinoline
methyl (2S,4R)-4-[2-(dimethyl-1,3-thiazol-4-yl)acetamido]-1-methylpyrrolidine-2-carboxylate
N-({1-[(2-cyanophenyl)methyl]piperidin-3-yl}methyl)-3-methylfuran-2-carboxamide
1-[4-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperazin-1-yl]ethan-1-one
4-benzyl-2-(hydroxymethyl)-N-(1-methyl-1H-pyrazol-4-yl)piperazine-1-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-ethyl-4-{[2-(1,4-oxazepan-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}-1H-pyrrole-2-carbonitrile
N-[(1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]-3-phenylpropanamide
8-[(4-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
3-(1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)propanoic acid
4-(5-methylpyridin-2-yl)-1-[4-(trifluoromethyl)pyridin-2-yl]piperidin-4-ol
3-({[(2-amino-1,3-thiazol-4-yl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-{5-[4-methoxy-3-(prop-2-en-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}pyridazine
3-(1H-imidazol-1-ylmethyl)-1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[1-(2-methylpropyl)cyclopropyl]amino}methyl)piperidin-2-one
N-[(3R,4S)-4-cyclopropyl-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{1'-[(1-propyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
(1S,5R)-6-(cyclopropylmethyl)-3-(5-phenyl-1,3,4-thiadiazol-2-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aR,7aS)-1-(2-methoxyacetyl)-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N,2-dimethyl-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide
(3R,4R)-1-[3-(4-fluorophenoxy)propyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
3-[(dimethylamino)methyl]-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-3-ol
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-benzyl-8-[2-(1H-pyrazol-1-yl)butanoyl]-2,8-diazaspiro[4.5]decan-3-one