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5-[(4-hydroxypiperidin-1-yl)methyl]-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
N-(1-hydroxybutan-2-yl)-3-methyl-1-propyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-4-carboxamide
2-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)azetidin-3-yl]pyridine
1-(2-{3-[(2-fluorophenyl)methoxy]phenyl}pyrimidin-4-yl)piperidin-3-ol
1-[1-(2-methylbenzoyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-3-fluoro-N-(oxolan-2-ylmethyl)benzamide
3-(1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carbonyl)pyridine
N-[(2-aminopyridin-3-yl)methyl]-6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[(E)-2-{3-[2-(oxolan-3-yl)-1H-imidazol-1-yl]phenyl}ethenyl]pyridine
N,1-dimethyl-N-[(3-{[1-(thiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperidin-4-amine
2-benzyl-N-[1-(thiophen-2-yl)propan-2-yl]-1,3-thiazole-4-carboxamide
[(4-ethyl-1,3-thiazol-2-yl)methyl]({[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl})amine
4-(1-ethyl-1H-imidazol-2-yl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidine
4-[3-ethoxy-4-(prop-2-en-1-yloxy)benzoyl]-3-methylpiperazin-2-one
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-(1,2-oxazinan-2-yl)propanamide
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(methoxymethyl)piperidine
1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(5-phenyl-1,3,4-thiadiazol-2-yl)urea
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
1-(4-methoxyphenyl)-3-methyl-4-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperazin-2-one
1-(cyclopropylmethyl)-4-(2,4-difluoro-3-methoxybenzoyl)-2-(propan-2-yl)-1,4-diazepane
2-ethyl-8-(5-methoxypyrimidin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]pyridine-3-carboxamide
6-cyano-N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyridine-3-carboxamide
2-(4-acetylphenoxy)-N-[2-(oxan-2-yl)ethyl]acetamide
2-amino-3-cyclopentyl-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propan-1-one
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-butyl-3-methyl-5-(trimethyl-1H-pyrazol-4-yl)-1H-1,2,4-triazole
N-methyl-2-(morpholin-4-yl)-N-(quinolin-5-ylmethyl)butanamide
N-[(3R,4S)-1-benzyl-4-cyclopropylpyrrolidin-3-yl]-2-methanesulfonamidoacetamide
1-[5-(dimethyl-1,2-oxazol-4-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
2-amino-4-{3-[1-(dimethylamino)ethyl]phenyl}-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
ethyl 1-(1H-1,2,3-benzotriazol-5-yl)-1H-imidazole-2-carboxylate
N-{[4-(dimethylamino)oxan-4-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-(2-methanesulfonylethyl)-4-propylpyrimidine-5-carboxamide
2-(2-ethylpyrimidin-5-yl)-7-methoxy-4-(morpholine-4-carbonyl)quinoline
1,3-dimethyl-2,4-dioxo-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]-1,2,3,4-tetrahydroquinazoline-6-sulfonamide
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]furan-2-carboxamide
4-(1-benzofuran-2-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(5-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridin-4-yl}-3-methyl-1H-1,2,4-triazol-1-yl)-6-methylpyridine
(3aS,6aS)-2-cyclohexyl-5-[2-(4-hydroxyphenyl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4R)-4-(dimethylamino)-1-({5-[(N-methylmethanesulfonamido)methyl]furan-2-yl}methyl)pyrrolidine-2-carboxylic acid
5-fluoro-2-[1-(morpholine-4-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
3-(3-methoxyphenyl)-4-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1H-pyrazole
(2R,6S)-2,6-dimethyl-4-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]morpholine
2-amino-4-(5-fluoro-2-methoxyphenyl)-6-(6-methoxypyridin-3-yl)pyridine-3-carbonitrile
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-{1-[1-(4-ethyl-5-methylpyrimidin-2-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(oxolane-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)oxane-2-carboxamide