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2-(cyclopropylmethyl)-9-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-6-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
(1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[2-(furan-2-yl)-2-oxoacetyl]piperidine-3-carboxylate
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3R,4R)-3-hydroxy-1-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperidin-4-yl]pyridine-2-carboxamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]quinoxaline-6-carboxamide
(1R,7S)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-4-oxo-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-cyclopropyl-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-(dimethylamino)-N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-fluorophenyl)acetamide
N-{2-methoxy-4-[2-methyl-3-(1H-pyrazol-1-yl)propanamido]phenyl}-3-methylbutanamide
3-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoic acid
2-(3-hydroxypropyl)-9-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(3aR,6aR)-2-(3-methylpyrazin-2-yl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2R)-2-amino-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-phenylacetamide
1'-(1,3-benzothiazole-6-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[(1R,2S)-2-phenylcyclopropyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-4-methanesulfonyl-1,4-diazepane
3-[(3R,4S)-4-(dimethylamino)-1-(2-propoxybenzoyl)piperidin-3-yl]propanoic acid
4-hydroxy-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
1-[(2,3-difluoro-4-methoxyphenyl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(3-methylpyridin-4-yl)methyl]-1H-pyrazole-3-carboxamide
3-ethyl-3-(hydroxymethyl)-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
1-phenyl-N-[2-(1,2,3-thiadiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]cyclopropane-1-carboxamide
N-cyclobutyl-2-(5-methyl-1,3-oxazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(2-cyclohexylethyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-4-yl]pyridine-3-carbonitrile
3-(4-methylpiperazine-1-carbonyl)-N-(prop-2-en-1-yl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
(3aR,6aR)-2-(3-chlorobenzoyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)-1H-pyrazole-3-carboxamide
5-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-methylpiperazine-1-sulfonamide
1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3-propoxypiperidine
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-1H-pyrazole-4-carboxamide
4-[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
1-(6-methyl-2-phenylpyrimidin-4-yl)-N-[(5-methylpyrazin-2-yl)methyl]piperidin-4-amine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
1-(4-hydroxy-4-phenylpiperidin-1-yl)-2-(1-methylpyrrolidin-2-yl)ethan-1-one
2-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-carbonyl}-N,N-dimethylaniline
3-[(1-acetylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]-4-methoxybenzamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-4-(pyrrolidin-3-yl)benzamide
3-{2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
N-[(3R,4S)-4-cyclopropyl-1-(oxan-4-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-5-carboxamide
3-[N-methyl4-(3-aminopiperidine-1-carbonyl)benzenesulfonamido]propanamide
3-ethyl-1-(3-methoxy-4-methylphenyl)-3-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]urea
2-ethyl-4-[4-(furan-2-yl)benzoyl]-1-(propan-2-yl)piperazine
4-[(3-chloropyridin-4-yl)methyl]-1-methylpiperazine-2-carboxylic acid