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4-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-methyl-1,4,9-triazaspiro[5.5]undecane
2-acetyl-N-[(5-methyl-2-{3-[3-(pyridin-3-yl)propanamido]phenyl}-1,3-oxazol-4-yl)methyl]benzamide
1-{2-[methyl({[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl})amino]ethyl}piperidin-2-one
2-{4-[4-(azocan-1-ylmethyl)phenoxy]piperidine-1-carbonyl}-1,3-benzothiazole
N-cycloheptyl-1-[2-(1H-indol-3-yl)ethyl]-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2,5-dimethylphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
N-[1-(4-chlorophenyl)ethyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[2-(2-fluorophenyl)-1-[1-(2-methylbutyl)piperidin-4-yl]ethyl]-N,2-dimethylfuran-3-carboxamide
N-(1-{7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
8-[2-(1H-imidazol-1-yl)acetyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-(1-carbamoylcyclopentyl)-3-(3-hydroxy-3-methylbutyl)benzamide
N-methyl-2-oxo-6-phenyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,2-dihydropyridine-3-carboxamide
1-[2-methoxy-5-(methylcarbamoyl)phenyl]-1H-imidazole-4-carboxylic acid
1-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-1-methyl-3-(5-phenyl-1H-1,2,4-triazol-3-yl)urea
(3S,4R)-1-[1-(3-methoxybenzoyl)piperidine-4-carbonyl]-4-methylpiperidine-3,4-diol
methyl 3-cyclobutaneamido-5-{[(3-methoxyphenyl)formamido]methyl}benzoate
4-(2,4-dioxoimidazolidin-1-yl)-N-(3-methyl-4-pentanamidophenyl)benzamide
N-methyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]-2,3-dihydro-1H-inden-2-amine
3-(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)pyridine
1-({1-[6-(benzylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-3-yl}methyl)pyrrolidin-2-one
N-(6-methoxy-2H-1,3-benzodioxol-5-yl)-2-methyl-3-oxo-4-phenylpiperazine-1-carboxamide
1-{7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(thiophen-3-yl)ethan-1-one
(2S,4R)-N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(thiophene-3-amido)pyrrolidine-2-carboxamide
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pentan-1-one
2-(dimethylamino)-N-[1-(hydroxymethyl)cyclohexyl]-2-(3-methylphenyl)acetamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}piperidin-3-ol
8-(7,8-dimethylquinolin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-amino-N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-phenylpyrimidine-5-carboxamide
N-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)methanesulfonamide
N6-benzyl-N5-methyl-N5-[3-(morpholin-4-yl)propyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]urea
N,N-dimethyl-3-[(2-oxo-4-phenylpyrrolidin-1-yl)methyl]-1,2,4-oxadiazole-5-carboxamide
2-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]-1H-imidazol-2-yl}-1-methyl-1H-imidazole
2-(3-oxo-9-{spiro[2.4]heptane-1-carbonyl}-2,9-diazaspiro[5.5]undecan-2-yl)acetamide
3-ethyl-5-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl]adamantan-1-ol
1-(morpholin-4-yl)-2-(4-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}phenoxy)ethan-1-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-(1,3-thiazol-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(4-{[4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,3-oxazol-2-yl]methyl}piperazin-1-yl)pyrimidine
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylprop-2-en-1-yl)acetamide
1-methyl-5-{[3-(methylsulfanyl)propyl]amino}-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,4S)-1-(1-benzoxepine-4-carbonyl)-4-[(2-hydroxyethyl)(methyl)amino]pyrrolidin-3-ol
N-cyclopropyl-N-[(4-hydroxyphenyl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1-(2-methylpropyl)piperidin-4-amine
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
N-(5-methyl-2,1,3-benzothiadiazol-4-yl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
(2R,3R,6R)-5-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-amino-N-methyl-N-[2-(oxan-2-yl)ethyl]-5,6,7,8-tetrahydroquinazoline-4-carboxamide
4-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid