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4-(3-chloro-4-hydroxy-5-methoxyphenyl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-4-(dimethylamino)butan-1-one
6-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-cyclopropylpyrimidin-4-ol
N-(2-hydroxyethyl)-5-(1-phenylcyclopropanecarbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-{2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
3-[(3S)-3-ethylmorpholin-4-yl]-N-(furan-2-ylmethyl)propanamide
(adamantan-1-ylmethyl)(methyl)(pyridin-3-ylmethyl)amine
8-(1-methyl-1H-pyrazole-3-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-cyclopropyl-2-(2-oxoazonan-1-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
4-[({[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]-2-methoxyphenol
6-cyclopentyl-1-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(2-fluorophenyl)methoxy]-8-(pyridin-2-ylmethyl)-1,8-diazaspiro[4.5]decan-2-one
2-[6-(2,3,4-trimethoxyphenyl)pyridin-3-yl]acetic acid
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-(hydroxymethyl)piperidin-3-ol
4-[(2-methoxyethyl)amino]-5-methyl-N-{[3-(trifluoromethoxy)phenyl]methyl}thieno[2,3-d]pyrimidine-6-carboxamide
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(1S,3R)-N1-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-1,2,N2,N3,3-pentamethylcyclopentane-1,3-dicarboxamide
methyl 3-({[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}carbamoyl)benzoate
N-{[1-(cyclopropanesulfonyl)-4-hydroxyazepan-4-yl]methyl}pyridine-3-sulfonamide
3-{[cyclopentyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)carbamoyl]methyl}-1,2,3-oxadiazol-3-ium-5-olate
5-methyl-5-phenyl-1-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}piperidin-2-one
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(1-phenylcyclopropanecarbonyl)piperidine
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(2-hydroxyethyl)piperidin-4-yl]methyl}acetamide
(2-{2-[1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
(1R,3S)-3-methoxy-7-[3-(piperidine-1-carbonyl)pyridin-2-yl]-7-azaspiro[3.5]nonan-1-ol
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}cyclopentanecarboxamide
3-({2-[1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-oxo-N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]butanamide
(5S,9aS,9bS)-5-(2,4-difluorophenyl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{1-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-4-yl}pyrimidin-2-amine
benzyl(cyclopropylmethyl){[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
(3S,4S)-1-(benzenesulfonyl)-4-[methyl(quinolin-5-ylmethyl)amino]pyrrolidin-3-ol
(3aR,6aR)-2-(6-ethyl-5-fluoropyrimidin-4-yl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(5-ethylthiophene-3-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2S,4S)-N,N-diethyl-4-(furan-3-amido)-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
N-{2-[1-(3-methylbut-2-en-1-yl)piperidin-3-yl]ethyl}piperidine-4-carboxamide
(2R,6R)-4-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-(2-hydroxyphenyl)-1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
9-[2-(pyrrolidin-1-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(3-methyl-1,2-oxazol-5-yl)acetamide
4-hydroxy-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
8-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3,5-dimethoxy-N-({1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-3-yl}methyl)benzamide
1-benzyl-3-[3-(pyridin-3-yl)propyl]-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamido-4-methylpentanamide
1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-phenylpiperazine
N-(1-benzothiophen-5-ylmethyl)-1-methyl-1H-pyrazole-5-carboxamide
1-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-amine
N-(2-methoxyethyl)-1-{1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
2-ethyl-9-{imidazo[1,2-a]pyridin-2-ylmethyl}-2,9-diazaspiro[5.5]undecan-3-one