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2-methoxy-4-[2-(pyridin-3-yl)piperidine-1-carbonyl]quinoline
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2-hydroxyethyl)-N-propyl-1,3-oxazole-4-carboxamide
5-(furan-2-carbonyl)-3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)pyridazine-4-carboxamide
3-({[(cyclopropylcarbamoyl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(methylsulfanyl)-1-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}ethan-1-one
6-({4-[3-(piperidin-1-yl)azetidine-1-carbonyl]-1,3-oxazol-2-yl}methoxy)quinoline
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-4-(4H-1,2,4-triazol-3-yl)piperidine
5-{2-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(4-methyl-1H-indazol-3-yl)phenol
{2-[4-(4-chlorophenyl)-2-methyl-5-oxopiperazin-1-yl]-2-oxoethyl}urea
N-benzyl-2-(4-fluorophenoxymethyl)-4-hydroxy-N-methylpyrimidine-5-carboxamide
5-methyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}thiophene-2-carboxamide
1,3-dimethyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-ethyl-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-chloro-N-(1,4-dioxan-2-ylmethyl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methylbenzamide
(3S,4S)-4-(dimethylamino)-1-[4-(3-hydroxy-3-methylbutyl)benzoyl]pyrrolidin-3-ol
4-[2-(4-fluorophenyl)ethyl]-11-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(5-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N-[3-({[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
({6,7-dimethoxy-2-[(4-methylphenyl)methoxy]quinolin-3-yl}methyl)[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-ethyl-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide
1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(pyridin-4-yl)propan-1-one
1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
3-(2-methoxyphenyl)-N-[(1R,3S)-3-(morpholine-4-carbonyl)cyclopentyl]propanamide
1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-(4-fluorophenyl)-N-[(4-hydroxyphenyl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
2-methyl-4-(4-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}phenyl)butan-2-ol
3-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
3-(2,3-dimethylquinoxalin-6-yl)-1-[2-methyl-1-(pyridin-2-yl)propyl]urea
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
2-(1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
4-acetyl-N-[1-(cyclohexylmethyl)piperidin-3-yl]benzamide
4-methyl-N-(2-methylpropyl)-3-(2-oxoimidazolidin-1-yl)-N-(pyridin-2-ylmethyl)benzamide
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
N-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-4-methyl-N-(oxolan-2-ylmethyl)benzamide
N-(1-hydroxy-3-methylbutan-2-yl)-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}butane-1,2-dione
(1S,5R)-3-(3-chloropyridin-2-yl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
9-{[6-(dimethylamino)pyridin-3-yl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[1-({[(8-methoxyquinolin-2-yl)methyl](methyl)amino}methyl)cyclopentyl]methanol
3-[1-(4-methylphenyl)cyclopentyl]-5-(pyrrolidin-1-ylmethyl)-1,2,4-oxadiazole
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
N-[(3-chloropyridin-4-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
1-(2H-1,3-benzodioxol-5-yl)-3-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}urea
N-benzyl-5-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)pyrimidin-2-amine
5-(4-methyl-1,4-diazepan-1-yl)-2-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydropyridazin-3-one
3-chloro-N-(2-methoxyethyl)-4-[(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)oxy]benzamide