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4-{5-[(2-chlorophenyl)methyl]-3-(ethoxymethyl)-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
(4S,4aS,8aS)-4-phenyl-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-decahydroquinolin-4-ol
N-(butan-2-yl)-2-(1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)benzamide
(4-{[2-(8-methoxyquinolin-2-yl)-1H-imidazol-1-yl]methyl}oxan-4-yl)methanol
diethyl({[3-(pyrrolidine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl})amine
N-[1-(butan-2-yl)-3-methyl-1H-pyrazol-5-yl]-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
N-[1-(3-methoxyphenyl)ethyl]-N-methyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
4-(3-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]oxy}benzoyl)morpholine
1-(2-methoxyethyl)-8-[(2-methyl-1H-indol-3-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{5-[(2S)-2-aminohexanamido]-2-methylphenyl}-3-methylbenzamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}propan-1-one
3-{[cyclopropyl(pyridin-2-ylmethyl)amino]methyl}-6-methoxy-1,2-dihydroquinolin-2-one
1-[1-(2-amino-5-butyl-6-methylpyrimidin-4-yl)piperidin-4-yl]piperidin-3-ol
N-cyclopropyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1S,7R)-2-methyl-4-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-4-azatricyclo[5.2.1.02,6]dec-8-ene-3,5-dione
N-({5-[(3-cyanophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
4-hydroxy-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine-4-carboxylic acid
1-[1-(4-fluorophenyl)cyclopropanecarbonyl]-3-(propoxymethyl)pyrrolidine
3-(oxolan-3-yl)-5-(1,2,5-trimethyl-1H-pyrrol-3-yl)-1,2,4-oxadiazole
3-[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]-1-azabicyclo[2.2.2]octane
1-[4-(furan-2-carbonyl)piperazin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
(3R,4S)-1-(4-methanesulfonylbenzoyl)-4-phenylpyrrolidin-3-amine
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(3-propyl-1H-pyrazole-5-carbonyl)-1,4-diazepan-5-one
4-{1-[(2-chlorophenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
1-({1-[2-methyl-2-(piperidin-1-yl)propyl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
N-{1-[1-(3-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]butyl}acetamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
(3R,4S)-4-cyclopropyl-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N,N-dimethylpyrrolidin-3-amine
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrazine-2-carboxamide
N-(1-{1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-cyclopropylpyridine-2-carboxamide
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-propyl-1H-1,2,4-triazol-3-amine
1-({4-methoxy-3-[3-(trifluoromethyl)phenoxy]phenyl}methyl)pyrrolidine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[(2R,6R)-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]ethan-1-one
(3S)-1-ethyl-3-methyl-4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
1-(2,6-dimethylpyridin-4-yl)-4-[4-(propan-2-yloxy)benzoyl]piperazine
1-(2,3-dihydro-1H-inden-2-yl)-4-[(pyridin-2-ylmethyl)amino]pyrrolidin-2-one
[(3R,4R)-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-(methylamino)pyridine-4-carboxamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-[(4-fluorophenyl)methyl]-1-(1-methyl-1H-pyrazole-4-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-[1-(cyclohexylmethyl)-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl]ethan-1-ol
(3S,4S)-4-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)pyrrolidine-3-carboxylic acid
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
(1R,9S)-5-amino-3-(1-benzofuran-2-yl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-{2-[(2,6-dichlorophenyl)methyl]-4-hydroxypyrimidine-5-carbonyl}piperidine-4-carbonitrile
9-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(2-fluoro-4-methoxyphenyl)methyl]-3-{2-oxo-2-[4-(pyrrolidin-1-yl)piperidin-1-yl]ethyl}piperazin-2-one
3-[3-({[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide