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2-{4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-1-yl}pyrimidine
(2S,4S)-4-amino-1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]pyrrolidine-2-carboxylic acid
4-[1-(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethyl]morpholine
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-3-amine
1-[3-oxo-3-(3-phenylpiperazin-1-yl)propyl]pyrrolidin-2-one
({5-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]furan-2-yl}methyl)dimethylamine
5-methoxy-9-[2-(1H-pyrazol-1-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecane
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[3-(methylsulfanyl)propyl]benzamide
2-methyl-3-{[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}quinoxaline
[3-(1H-pyrazol-1-yl)propyl]({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
N-[2-hydroxy-1-(pyridin-3-yl)ethyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
3-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3,9-diazaspiro[5.6]dodecan-10-one
4-{4-[(1-methyl-1H-indol-6-yl)methyl]piperazin-1-yl}quinazoline
4-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-{2-[1-(2-cyclopropyl-1,3-benzoxazole-6-carbonyl)piperidin-2-yl]ethyl}phenol
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[(6-methylpyridin-2-yl)methyl]acetamide
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea
4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-phenylpiperazin-2-one
N,2,7-trimethyl-N-[2-(oxan-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3R,9aR)-3-(hydroxymethyl)-8-[(4-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(2-ethyl-1H-imidazol-1-yl)propanamide
2-{1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}acetic acid
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-(1,3-benzothiazol-2-yl)-4-[(1-methylpyrrolidin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(2S)-1-(4-{[(2-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidin-2-yl]methanol
2-{2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-2-oxoethyl}-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
1-{8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
1-cyclopropyl-N-[3-(2-methoxyphenyl)propyl]-6-oxopiperidine-3-carboxamide
1-cyclohexyl-4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-methyl-2-{3-oxo-2-azaspiro[4.5]decan-2-yl}-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
N-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-N-(2-phenylethyl)acetamide
N-{[1-(5-ethyl-1,3,4-thiadiazol-2-yl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
2-benzyl-9-(2-hydroxypropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(cyclohexylmethyl)-5-[(3-hydroxypropyl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{5-cyclopropyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(2,5-dimethoxyphenyl)pyrimidine
3-{5-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]propanamide
(3S,4S)-4-(4-fluorophenyl)-1-(3-methyl-1H-pyrazole-4-carbonyl)piperidin-3-ol
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-1-yl}-1,3-benzothiazole
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
5-amino-N-methyl-N-[(1-methylpiperidin-3-yl)methyl]-4-phenyl-1H-pyrazole-3-carboxamide
4-[4-(1-cyclopropanecarbonylpiperidine-4-carbonyl)piperazin-1-yl]-5,6-dimethylpyrimidine
(1,3-benzoxazol-2-ylmethyl)({[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-[1-(pyridin-3-yl)propan-2-yl]-6-azaspiro[2.5]octane-1-carboxamide
1-(4-benzylpiperidin-1-yl)-3-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-4-yl]propan-1-one
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-3-(pyridin-4-yl)propan-1-one