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(1R,5R)-N,N-dimethyl-6-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-phenyl-1-[1-(thiophen-3-ylmethyl)piperidin-3-yl]propan-1-one
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-2,3-dimethyl-N-(pyridin-4-ylmethyl)-1H-indole-5-carboxamide
3-chloro-N-[2-(4-ethylphenoxy)ethyl]-N-methylpyridine-4-carboxamide
1-{2-[1-(2-methoxy-6-methylbenzoyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
(2S,4S)-4-amino-N-ethyl-1-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]pyrrolidine-2-carboxamide
(1R,2S)-N-methyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]cyclohexane-1-carboxamide
2-(3-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
1-{2-[methyl({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl})amino]pyrimidin-4-yl}piperidin-4-ol
2-{1-[2-(pyridin-3-yl)-1,3-benzoxazol-5-yl]-1H-pyrazol-4-yl}ethan-1-ol
1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-phenylpropan-1-one
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(3-fluorophenoxy)ethan-1-one
1-(1-{[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
(1S,5R)-6-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(6-methylpyridazin-3-yl)-decahydro-1,6-naphthyridin-2-one
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-2,4-dimethylpyrimidine
3-(5-cyclopropyl-3-methyl-1H-pyrazol-4-yl)-N,N-dimethylbenzamide
1-[(3-methylpyridin-2-yl)methyl]-4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazine
[4-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)morpholin-3-yl]methanol
2-(3-methoxypropyl)-8-[5-(propan-2-yl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
1-cyclopentyl-4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidin-3-amine
1-{imidazo[1,2-a]pyridine-3-carbonyl}-3-(3-methoxyphenoxymethyl)piperidine
4-[2-(3,5-dimethylpiperidin-1-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
8-{2-methylthieno[2,3-d]pyrimidin-4-yl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-(1-{1-[(4-chlorophenyl)methyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl}ethyl)methanesulfonamide
1-{2-oxo-2-[(2S)-2-(piperidine-1-carbonyl)pyrrolidin-1-yl]ethyl}-1,2,3,4-tetrahydroquinolin-2-one
2-{4-[(3-ethoxy-4-methoxyphenyl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
(3S,4R)-4-(3-methoxyphenyl)-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]pyrrolidine-3-carboxylic acid
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(1H-imidazol-2-ylmethyl)piperidine
1-{3-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}propan-1-one
3-(3-methoxyphenyl)-1-phenyl-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
benzyl(butyl){[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
(1R,5R)-6-[4-(difluoromethoxy)benzoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[4-(thiophen-2-yl)butanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-(2,4,5-trimethoxybenzoyl)pyrrolidin-3-yl]methanol
3-(2-ethyl-1H-imidazol-1-yl)-1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
2-[(4aR,8aR)-7-cyclobutanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-N-benzylacetamide
2-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluorophenyl)ethyl)piperidin-1-yl]methyl}-3-methoxyphenol
2-(2-methoxyethoxy)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]ethan-1-one
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(9H-purin-6-yl)-2,8-diazaspiro[4.5]decan-3-one
3-methyl-3-[2-(methylsulfanyl)ethyl]-1-(3,4,5-trimethoxyphenyl)urea
3-acetyl-N-[(3R,4R)-3-hydroxypiperidin-4-yl]benzamide
2-[4-(benzyloxy)piperidine-1-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
5-acetyl-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]thiophene-2-carboxamide
4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}benzamide
4-[2-(2-methoxyethoxy)acetyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
3-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one