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N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-6-methoxypyrimidin-4-amine
2-[2-(2-methoxy-4-methylphenyl)-1H-imidazol-1-yl]propan-1-ol
4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-(propan-2-yloxy)pyrimidin-2-amine
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-(1-methylpiperidin-2-yl)propanamide
N-methyl-2-(methylsulfanyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-N,4-dimethylaniline
1-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-cyclopropylethan-1-one
(1-{[1-(2-ethylbutyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-phenylpiperidine-1-carboxamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-4-ylmethyl)pyridin-2-amine
4,6-dimethyl-2-[4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-1-yl]pyridine-3-carbonitrile
N-(cyclopropylmethyl)-N-propyl-2-(thiophene-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-(1H-indol-4-ylmethyl)benzamide
N-[(1-hydroxycyclohexyl)methyl]-3-(1H-pyrazol-4-yl)benzamide
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-(pyridin-3-yl)piperazine
N-[5-(6-hydroxy-4-methyl-1,4-diazepane-1-carbonyl)-1,3-thiazol-2-yl]acetamide
N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
N4-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N4-methyl-5,6,7,8-tetrahydroquinazoline-2,4-diamine
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-3-propanamidobenzamide
7-methyl-2-[4-(2-oxopyrrolidin-1-yl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
5-[1-(6-hydroxypyridine-3-carbonyl)pyrrolidin-2-yl]-N-(pyridin-3-yl)thiophene-2-carboxamide
1-[(2-chloro-4-hydroxyphenyl)methyl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
4-{[2-(dimethylamino)-6-methylpyrimidin-4-yl]amino}-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-[3-(propan-2-yloxy)benzoyl]piperidine
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(4-methoxyphenyl)methyl]piperidine
5-(2,4-difluorophenoxymethyl)-N-(2-hydroxyethyl)-N-methyl-1,2-oxazole-3-carboxamide
5-[(methylsulfanyl)methyl]-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-[2-(3-fluorophenyl)ethyl]-N-(2-methylprop-2-en-1-yl)-6-oxopiperidine-3-carboxamide
1-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-3-(hydroxymethyl)pyrrolidin-3-ol
3-amino-1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-hydroxypropan-1-one
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[(3R,4S)-1-cyclopentyl-4-propylpyrrolidin-3-yl]acetamide
9-(2-phenylbenzoyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-(3-cyclohexylpyrrolidin-1-yl)-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-2-(methylsulfanyl)acetamide
(2S,4R)-4-amino-1-(6-cyclopropylpyrimidin-4-yl)-N-ethylpyrrolidine-2-carboxamide
1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-[3-(trifluoromethyl)benzoyl]piperidine
1-{4-[2-(3,4-dimethoxyphenyl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-3-amine
(2S,4S)-4-amino-N-(propan-2-yl)-1-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]pyrrolidine-2-carboxamide
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methyl-1,3-oxazole-5-carboxamide
5-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperazine-1-sulfonamide
N-methyl-4-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-thiazol-2-amine
N-(furan-2-ylmethyl)-2-(hydroxymethyl)-N-(thiophen-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
3-[(2R,3R,6R)-5-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-({[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl](methyl)amino}methyl)-3,4-dihydroquinazolin-4-one
1-(4-chlorophenyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]cyclobutane-1-carboxamide