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4-(1-butyl-1H-imidazol-2-yl)-1-[(4-methylthiophen-2-yl)sulfonyl]piperidine
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-propanoylpiperidine-4-carboxamide
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
2-(1-butyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}acetamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
2-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydro-1,2-benzothiazol-3-one
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-2-one
9-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridine
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2-methyl-1-benzofuran-5-carboxamide
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3-(thiophen-2-yl)propanamide
N-methyl-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}-3-propanamidobenzamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-4-(piperidin-1-yl)butanamide
3-(1,2-oxazinan-2-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide
4-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
7-(3-chlorophenyl)-4-[(2-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-2-ethyl-2,5-dihydro-1H-pyrrole-1-carboxamide
5-phenyl-3-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-1,2-oxazole
(1R,5S,8R)-3-({3-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)-3-azabicyclo[3.2.1]octan-8-ol
1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
2-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,3-thiazole
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
6-[(3R,4R)-3-hydroxy-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-1-yl]pyridine-2-carbonitrile
3-(2-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-4-[(4-methylphenyl)methyl]piperazin-2-one
2-cyclopentyl-N-[3-(4-{[(4-phenyl-1,3-thiazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
N-(2-methoxyphenyl)-2-{3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
(1R,3S)-3-(2-aminoethoxy)-7-(5-chloro-1H-indole-2-carbonyl)-7-azaspiro[3.5]nonan-1-ol
1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-2-(2-methylphenyl)pyrrolidine
8-cyclopentyl-3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(6-methylpyridin-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-6-(quinolin-8-yl)pyridazin-3-amine
3-[2-(5-phenylthiophen-2-yl)-1H-imidazol-1-yl]propanamide
1-(azocan-1-yl)-3-[5-({[(4,6-dimethylpyrimidin-2-yl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-(cyclohex-3-en-1-ylmethyl)-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N-(4-tert-butylphenyl)-4-(9H-purin-6-yl)piperazine-1-carboxamide
6-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)cyclopentanamine
N-[(2-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-(1H-1,2,4-triazol-5-yl)benzamide
N-(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-(4-fluorophenyl)piperidin-4-ol
N-(3-methoxyphenyl)-3-{1-[(3-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}propanamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-({7-[(2,3-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-(3-fluorophenyl)acetamide
1-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[4-(4-methylpiperazin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
2-{[4-(4-fluoro-2-methylphenyl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
2-{4-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-N-ethylacetamide