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1,9-dimethyl-4-{[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl}-1,4,9-triazaspiro[5.5]undecane
2-{2-methylthieno[3,2-d]pyrimidin-4-yl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
methyl 6-[(4-acetylpiperazin-1-yl)methyl]-3-benzamidothieno[2,3-b]pyridine-2-carboxylate
2-[4-(8-methoxy-2-methylquinolin-5-yl)-3,5-dimethyl-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1-(4-fluorobenzoyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(propyl)(pyridin-4-ylmethyl)amine
[(3R,4R)-1-(2-chloro-6-fluoro-3-methylbenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-cyclopropylethan-1-one
4-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
1'-hexyl-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-4-{[(2,4-difluorophenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
5-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexane-3-carbonyl]-2-methylphenol
2-methoxy-N-methyl-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]pyridine-4-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2-methyl-1H-indol-3-yl)acetamide
1-(2-phenylethyl)-4-[1-(1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]piperidine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1H-imidazole-2-carboxamide
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-2-(ethylamino)pyrimidine-5-carboxamide
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,1-benzoxazole-3-carboxamide
1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-3-ol
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-{methyl[(4-methylphenyl)methyl]amino}ethan-1-one
(4aS,8aR)-6-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-1-(2-methylpropyl)-decahydro-1,6-naphthyridin-2-one
4-chloro-N-(1H-imidazol-2-ylmethyl)-N-methyl-2-propanamidobenzamide
{3-[(dimethylamino)methyl]-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)piperidin-3-yl}methanol
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
5-(methoxymethyl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)furan-2-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[3-(3-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-(prop-2-en-1-yl)butanamide
4-[3-(benzyloxy)propyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
N-(1H-indol-3-yl)-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-[3-(trifluoromethyl)phenyl]acetamide
(1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)methanol
4-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
N-methyl-N-(pyridin-3-ylmethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
4-cyclopropyl-1-(2-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-oxoethyl)-4-methylpyrrolidin-2-one
3-(1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
2-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]propane-1,3-diol
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-methyl-N-(oxan-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-{1-[7-(cyclohexylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}acetamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}piperidine
8-(7-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1,3-benzothiazole-6-carboxamide
7,7-dimethyl-2-{[(1-methyl-1H-imidazol-2-yl)sulfanyl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carbonitrile
1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
[5-(2,6-dimethoxyphenyl)-1H-1,3-benzodiazol-2-yl]methanol
4-(2,6-dimethylpyridin-3-yl)-N-[(5-ethylpyridin-2-yl)methyl]-N-methylpyrimidin-2-amine
4-(4-chlorophenoxy)-N-(2-hydroxy-2-phenylethyl)piperidine-4-carboxamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N-benzyl-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide