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N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(3-hydroxyquinoxalin-2-yl)propanamide
N,6-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-4-[4-(methylsulfanyl)phenyl]-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(1-{[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-(3-fluorobenzoyl)-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
2-amino-6-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-4-(piperidin-4-yl)pyridine-3-carbonitrile
N-benzyl-N-methyl-3-{[(1-phenylethyl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
ethyl 4-(oxan-2-ylmethyl)-1-[(2-phenylethyl)carbamoyl]piperidine-4-carboxylate
5-ethyl-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
2-{3-methyl-5-[(2,2,3,3-tetrafluoropropoxy)methyl]-1H-1,2,4-triazol-1-yl}benzoic acid
4-{[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]methyl}-3-(3,4,5-trimethoxyphenyl)-1H-pyrazole
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-1-(3-methylbutyl)-1H-pyrazole
3-(2-methoxyphenyl)-N-{2-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}propanamide
2-{5-cyclopropyl-4-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}-4-(5-methylfuran-2-yl)pyrimidine
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[(3,4,5-trimethoxyphenyl)methyl]acetamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
1,3-dimethyl-6-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(2E)-3-phenylprop-2-en-1-yl]-4-(piperidine-3-carbonyl)piperazine
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[2-(pyridin-3-yloxy)ethyl]-1H-pyrazole-4-carboxamide
6-{2-[5-(oxolan-2-yl)thiophen-2-yl]-1H-imidazol-1-yl}-1H-indazole
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-(4-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
[(6-methoxy-1H-indazol-3-yl)methyl](methyl)(quinolin-5-ylmethyl)amine
1-(1-methyl-1H-imidazole-2-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[(3R,4S)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-cyclopropylpyrrolidin-3-yl]-3-hydroxypropanamide
4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-methylquinoline
N-{[1-(cyclohex-2-en-1-yl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}-3-methoxybenzamide
4-(1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)benzoic acid
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-1-{2-[1-(5-fluoro-2-methylbenzenesulfonyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
3-[1-(1H-indole-6-carbonyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
4-ethyl-5-methyl-6-[3-(pyrimidin-4-yl)piperidin-1-yl]pyrimidin-2-amine
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-2H-1,3-benzodioxole-5-carboxamide
(3S,4S)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine-3,4-diol
1-cyclohexyl-4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazine
N-(propan-2-yl)-1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-(3-{[4-(isoquinolin-1-yl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
4-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carbonyl}-1,4-oxazepane
N-{1-[7-(2-ethylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-phenylpropanamide
4-ethyl-3-{1-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-2-[4-(morpholin-4-yl)-2-[(2-phenylethyl)amino]pyrimidin-5-yl]propanoic acid
4-(1-ethyl-1H-imidazol-2-yl)-1-[4-(2-methoxyphenyl)benzoyl]piperidine
N-ethyl-3-methyl-5-propyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1-benzofuran-2-carboxamide
2-[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]-6-methylpyridine-3-carbonitrile
1-cyclopentyl-4-({[1-(2-methylpropyl)piperidin-4-yl]amino}methyl)pyrrolidin-2-one
N-[4-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)-4-oxobutyl]acetamide
8-(4-propylpyrimidine-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-cyclopropyl-N-[2-(naphthalen-1-yl)propan-2-yl]-6-oxopiperidine-3-carboxamide
2-[1-(3-methylbut-2-en-1-yl)-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperazin-2-yl]ethan-1-ol
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[1-(4-methylphenyl)propyl]propanamide