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4-[1-(1H-imidazol-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]benzoic acid
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N,5-dimethyl-1,3-oxazole-4-carboxamide
N-({2-[4-(pyrrolidine-1-sulfonyl)phenyl]phenyl}methyl)propanamide
4-[2-(3-phenylpyrrolidin-1-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-{2-methyl-5-[3-(pyridin-3-yl)azetidine-1-carbonyl]phenyl}imidazolidin-2-one
N-methyl-2-(4-methyl-1H-pyrazol-1-yl)-N-{[3-(methylsulfanyl)phenyl]methyl}propanamide
1-[1-ethyl-5-(4-methylbenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]pyrrolidine
3-amino-1-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-[(1-ethylpiperidin-3-yl)methyl]-N-methyl-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-(4-fluorophenyl)piperidine
1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-3-phenylbutan-1-one
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-[2-(2,4-difluorophenyl)-1-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}ethyl]-N-methylpyridine-3-carboxamide
N-(5-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}pyrimidin-2-yl)benzenesulfonamide
1-(2,3-dihydro-1H-indol-1-yl)-2-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
N,N-dimethyl-5-[1-(quinolin-3-ylmethyl)-1H-1,2,3-triazol-4-yl]pyridin-2-amine
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-[4-(3-methylpiperidin-1-yl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
7-hydroxy-6-methyl-4-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-1,2,3,4-tetrahydroquinolin-2-one
N-[2-(1-benzylpiperidin-3-yl)ethyl]oxane-4-carboxamide
methyl (2S,4S,5R)-4-[(cyclopropylmethyl)carbamoyl]-5-(2-fluorophenyl)-1-methylpyrrolidine-2-carboxylate
5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-cyclohexylurea
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-hydroxyphenyl)ethan-1-one
2-[4-({methyl[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenyl]-6-phenyl-3,4-dihydropyrimidin-4-one
2-phenyl-1-[1-(thiophene-3-sulfonyl)piperidin-3-yl]ethan-1-one
{4-[(1-cyclobutanecarbonylpyrrolidin-3-yl)methyl]phenyl}methanol
3-({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)propanamide
methyl 3-[2-(2,3-difluorophenyl)acetyl]-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[ethyl({[(3R,4R)-1-(5-fluoro-2-methylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
N-ethyl-3-(2-hydroxy-2-methylpropanamido)-N-phenylbenzamide
8-[(5-carboxy-1-methyl-1H-pyrrol-2-yl)sulfonyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(propan-2-yl)-2-({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)acetamide
2-cyclopropyl-8-(2,6-difluorobenzenesulfonyl)-2,8-diazaspiro[5.5]undecan-3-one
7-methoxy-N-[3-(pyridin-4-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[3-(methylsulfanyl)propyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
N3-[1-(furan-2-yl)ethyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
[3-(2-phenoxyethyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-3-yl]methanol
1-[(4aR,8aR)-7-[2-(dimethylamino)benzoyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
N-(3-cyclopentylpropyl)-5-(2,6-difluorophenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
N-{[7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]pyridine-3-carboxamide
3-[(4-fluorophenyl)methyl]-1-(3-fluoropyridin-2-yl)piperidine-3-carboxylic acid
4-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)-1-propylpyrrolidin-2-one
3-cyclopentyl-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
2-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[(3-methyloxetan-3-yl)methyl]-1H-pyrazole-3-carboxamide
4-{[1-(1,3-dihydroxypropan-2-yl)pyrrolidin-3-yl]methyl}benzoic acid
N,2-dimethyl-4-oxo-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indole-3-carboxamide