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(1S,5R)-6-(cyclopropylmethyl)-3-(quinoline-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
[(3R,4R)-1-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-{2-oxo-2-[3-(pyridine-2-carbonyl)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
N3-(1,3-benzothiazol-2-ylmethyl)-N5-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]-1H-imidazole-4-carboxylic acid
N-({5,7-dimethylimidazo[1,2-a]pyridin-2-yl}methyl)-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
5-(2,3-dihydro-1-benzofuran-2-carbonyl)-3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-({5-[(2,5-dimethylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-6-methoxyhexanamide
N-[3-(1H-imidazol-1-yl)propyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amine
3-(6-methyl-2-propylpyrimidin-4-yl)phenol
1-{1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]piperidin-4-yl}-2-phenylethan-1-ol
1-{1-[(4-cyanophenyl)methyl]piperidin-4-yl}-N-cyclopropylpiperidine-3-carboxamide
N-ethyl-N-(2-hydroxyethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
3-(2-ethoxybutyl)-1-(2-fluoro-4-methylphenyl)urea
2-(2-methyl-1H-indol-3-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
N-butyl-2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-[(2-methylphenyl)methyl]acetamide
N-[(1R,2R)-2-hydroxycyclohexyl]-2-(phenylamino)-N-propylpyrimidine-5-carboxamide
5-{[methyl(2-phenylethyl)amino]methyl}-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
3-ethyl-N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-1H-indole-2-carboxamide
4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3-(3-methoxyphenyl)-1H-pyrazole
N,N-diethyl-1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carboxamide
3-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-[5-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]piperidine
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-methylimidazo[1,2-a]pyridine-2-carboxamide
6-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(1H-1,3-benzodiazol-1-yl)-N-(isoquinolin-5-ylmethyl)-N-methylpropanamide
5-{[benzyl(methyl)amino]methyl}-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
1-{2-[3-(pyridin-2-yl)azetidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
1-{[3-(cyclopentyloxy)phenyl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(9aR)-8-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[3-(3-methoxypropyl)piperidin-1-yl]pyridine-4-carboxamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
N-ethyl-3-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}propanamide
1-{2-[1-(2-fluoro-6-methoxybenzoyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
6-(propan-2-yloxy)-N4-(pyridin-3-ylmethyl)pyrimidine-2,4-diamine
6-[(diethylamino)methyl]-N-[4-(hydroxymethyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(2S,4S)-N-ethyl-1-[(4-ethylphenyl)methyl]-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
8-{[2-(furan-2-yl)phenyl]methyl}-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1,3-diphenyl-1H-pyrazole-5-carbonyl)azepan-4-amine
1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazole
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridin-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
3-(3-ethylphenoxy)-1-[(2R)-oxolane-2-carbonyl]azetidine
1-(morpholin-4-yl)-3-[1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)piperidin-3-yl]propan-1-one
1-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-N-cyclopropylpiperidine-4-carboxamide
3-{1-benzyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-4-chloro-1-methyl-1H-pyrazole
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-chloro-5-(methylcarbamoyl)phenyl]-4-(6-methylpyridin-2-yl)piperazine-1-carboxamide