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N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
2-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)pyrrolidin-3-yl]benzoic acid
6-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidine-1-carbonyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-(1,2,4-oxadiazol-3-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine
1-{4-[2-(phenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
2-(4-fluorophenyl)-N-(2-{7-[(5-methylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-[3-(trifluoromethyl)benzoyl]piperidine
3-[1-(1-benzyl-5-methyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-({2-[methyl(phenyl)amino]propyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-2-hydroxy-4-(methylsulfanyl)butanamide
N-[(2-methylphenyl)methyl]-4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
2-({2-[cyclopentyl(methyl)amino]acetamido}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(prop-2-en-1-ylsulfanyl)ethan-1-one
6-(aminomethyl)-2-[4-({[2-(dimethylamino)-1-phenylethyl](methyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-(1-{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
1-[(3S)-3-(dimethylamino)azepan-1-yl]-2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[2-(methylsulfanyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(4-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-oxobutyl)acetamide
2,3-dimethyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]quinoxaline-6-carboxamide
5-(2-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}-2-oxoethyl)-1,3-dimethylimidazolidine-2,4-dione
(1R,7S)-N-methyl-4-oxo-3-[4-(propan-2-yl)phenyl]-N-[2-(1H-pyrazol-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-(5-methoxypyridin-3-yl)quinoxaline
3-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-N-(pyridin-4-yl)benzamide
N-(2-methoxyethyl)-5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[4-(thiophen-2-yl)butanoyl]piperidine-4-carboxamide
(3S,5R)-5-(2,3-dihydro-1H-isoindole-2-carbonyl)-N-(6-methylpyridin-3-yl)piperidine-3-carboxamide
(5S)-5-{[benzyl({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]methyl}pyrrolidin-2-one
2-amino-8-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
3-(1-methyl-1H-pyrazol-4-yl)-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethyl-1H-pyrrole-3-carboxamide
(3S,9aR)-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2,3-dimethyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(5-methyl-1H-indazole-3-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[cyclohexyl(methyl)amino]-3-[2-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
4-{5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(2-fluoroethyl)benzamide
4-(1-benzoylpiperidin-4-yl)-N-cyclopropylpiperazine-2-carboxamide
9-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-[2-(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]morpholine
(1R,5S)-8-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,8-diazabicyclo[3.2.1]octane
1-[4-({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,4-diazepan-1-yl]-2-methoxyethan-1-one
1-(2-{1-[2-(2,4-dimethoxyphenyl)acetyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
4-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
8-methyl-2-(pyrimidin-5-yl)-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)quinoline
N-{4-[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]-2-methoxyphenyl}acetamide
7-cyclohexyl-2-(1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)propanamide
N-(isoquinolin-5-ylmethyl)-N,2-dimethyl-4-phenylpyrimidine-5-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{2-[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrazine
7-[(3-methoxyphenyl)methyl]-2-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2,7-diazaspiro[4.5]decane