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(2S,4S)-4-amino-1-[3-(3,4-dimethoxyphenyl)propanoyl]pyrrolidine-2-carboxylic acid
2-(2-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-4-(pyrimidin-2-yl)phenoxy)acetic acid
2-(4-{[ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenoxy)ethan-1-ol
methyl(1H-pyrazol-3-ylmethyl)[(2,3,6-trifluorophenyl)methyl]amine
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
methyl 2-[4-(1,3-benzothiazole-6-carbonyl)-2-oxopiperazin-1-yl]acetate
3-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-ethylpropanamide
(1S,5R)-6-(1,3-dimethyl-1H-indole-2-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(3aS,6aS)-2-cyclopentanecarbonyl-5-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3R,4R)-1-(2-methoxy-6-methylbenzoyl)-3,4-dimethylpyrrolidin-3-ol
7-fluoro-4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-2-methylquinoline
4-hydroxy-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-(3-methyl-1H-pyrazole-5-carbonyl)-1,4-diazepane
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-ethyl-N-(2-methoxyethyl)pyridin-2-amine
6-(2,3-dihydro-1H-inden-2-yl)-1-(4-methyl-1,4-diazepane-1-carbonyl)-6-azaspiro[2.5]octane
N-(2-hydroxyethyl)-3-{5-[(3-hydroxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
3-(1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-N-phenylpropanamide
6-{4-[(3-methyl-1-benzothiophen-2-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
N-butyl-2-{methyl[2-(morpholine-4-carbonyl)pyridin-4-yl]amino}acetamide
(1S,5R)-3-[(2-butyl-1H-imidazol-4-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(2-{1-[3-(2-oxoazepan-1-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
[1-ethyl-5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
5-[2-(cyclohexylamino)pyrimidin-4-yl]-2-ethoxybenzoic acid
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1-(propan-2-yl)piperidine-3-carboxamide
2-(3-{8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}piperidin-1-yl)acetamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
(1R,5R)-3-(3,5-dichloro-4-methylbenzoyl)-3,9-diazabicyclo[3.3.2]decan-10-one
4-{5-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1H-pyrazol-3-yl}pyridine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[2-(phenylsulfanyl)ethyl]-3,6-diazabicyclo[3.2.2]nonane
N-{2-[2-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-1,3-thiazol-4-yl]ethyl}thiophene-2-carboxamide
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(1H-indazol-1-yl)acetamide
N-{1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-4-yl}methanesulfonamide
(3R,4R)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
N-[(2,3-dimethylphenyl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
N-(4-fluoro-2-methylphenyl)-2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamido]propanamide
8-{[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}quinoline
2-(3-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}phenoxy)ethan-1-ol
N-[2-(5-chloro-2-methyl-1H-indol-3-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-(2,2-diphenylethyl)-2-(2-oxopyrrolidin-1-yl)acetamide
2-{1-[4-(4-fluorophenyl)oxane-4-carbonyl]pyrrolidin-2-yl}pyridine
4-(3-methanesulfonylpropanoyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
3-hydroxy-3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
6-[3-(aminomethyl)pyrrolidin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
1-(4-fluorophenyl)-2,2-dimethyl-N-[3-(morpholin-4-yl)propyl]cyclopropane-1-carboxamide
2-methyl-6-[3-(4-phenylbenzoyl)piperidine-1-carbonyl]pyridine
3-(4-methyl-1,3-thiazol-5-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
5-acetyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]thiophene-3-carboxamide
ethyl 2-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)acetate
1-(4-methanesulfonyl-1,4-diazepan-1-yl)-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one