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1-[3-(1H-imidazol-2-yl)benzoyl]-3,4,4-trimethylpyrrolidin-3-ol
5-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)thiophene-2-sulfonamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}piperidin-2-one
N-[1-(pyrazin-2-yl)piperidin-3-yl]-1H-pyrazole-4-carboxamide
6-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
1-cyclohexyl-N-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
4-(1H-indol-4-yl)-3-phenyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(2-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-[(3-methyl-7-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]thiophene-3-carboxamide
(2R,6S)-4-(1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-2,6-dimethylmorpholine
2-(2-hydroxyethyl)-6-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
4-[1-(2-phenylethyl)piperidin-4-yl]-6-(pyrrolidin-1-yl)pyrimidine
methyl 3-(5-methylpyrazine-2-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
ethyl 5-benzyl-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
{[3-(4-chlorophenoxy)phenyl]methyl}(methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
1-(5-chloropyridin-2-yl)-4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-3-yloxy)piperidine-1-carboxamide
2-(5-methyl-1,2-oxazol-3-yl)-1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidine
methyl 2-(ethylsulfamoyl)-6-(1-phenylcyclopropanecarbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-2-[(dimethylamino)methyl]-1,3-thiazole-4-carboxamide
(4aR,7aS)-1-{2-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-8-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-oxo-1-[(3-phenyl-1H-pyrazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
N-{[5,8-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
2-{4-[6-(propan-2-yl)pyrimidin-4-yl]morpholin-2-yl}ethan-1-amine
1-(3-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}piperidin-1-yl)propan-1-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-1-methyl-6-oxo-N-(pyridin-3-ylmethyl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-cyclopentyl-N-[1-(4-fluorophenyl)piperidin-4-yl]-5-oxopyrrolidine-3-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(propane-2-sulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(1-benzofuran-2-ylmethyl)-3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-(methylsulfanyl)-3-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridine
3-[2-(dimethylamino)ethyl]-3-(oxolan-2-ylmethyl)-1-[3-(pyridin-3-yl)phenyl]urea
2-({4-cyclopentyl-1-[(4-methoxyphenyl)methyl]-2-oxo-1,4-diazepan-6-yl}oxy)-N,N-diethylacetamide
2-({ethyl[(3R,4R)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]amino}methyl)benzoic acid
4-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]thiomorpholine
N-[2-(1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethyl]acetamide
1-[(4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)methyl]piperidine
N-(4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenyl)acetamide
5-cyclohexaneamido-N-[2-(diethylamino)ethyl]-N-ethyl-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
3-{[(5-methylpyrazin-2-yl)methyl]amino}-N-(pyridin-3-yl)propanamide
1-(1-benzofuran-3-carbonyl)-4-(hydroxymethyl)azepan-4-ol
N,N-dimethyl-3-[4-(pyridin-4-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
1-{5-[(4-cyclopentylpiperazin-1-yl)methyl]-2-methoxyphenoxy}-3-(piperidin-1-yl)propan-2-ol
4-[5-(2-phenyl-1H-imidazol-1-yl)furan-2-carbonyl]morpholine
methyl 3-acetamido-5-{[(3-hydroxyphenyl)methyl]amino}-1-[2-(1H-indol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-ethyl-2-methoxy-3-({[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}methyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-(methanesulfonylmethyl)-1-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidine