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{1-[1-(2-ethoxybenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methanol
N-(pyridin-2-ylmethyl)-2-[4-(1H-1,2,4-triazol-1-yl)butanamido]benzamide
4-[(2-fluorophenyl)methyl]-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
1-benzyl-8-[(4-hydroxyphenyl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-ethyl-N-methyl-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-[2-(1-methyl-1H-pyrazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-1-phenylcyclopropane-1-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
N-[(2R,3R)-2-hydroxy-1'-(isoquinolin-5-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
2-({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
N-methyl-5-(morpholin-4-ylmethyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]furan-3-carboxamide
N-ethyl-1,3-dimethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-(2H-1,3-benzodioxol-5-yl)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methylpropanamide
5-cyclobutyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3,4-oxadiazol-2-amine
9-{[3-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N,6-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}quinolin-4-amine
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-2-acetamidoacetamide
2-acetyl-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
(2H-1,3-benzodioxol-4-ylmethyl)[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amine
1-(3-methylpyridin-2-yl)-4-(pyrrolidin-3-ylmethyl)piperazine
1-[(3-hydroxyphenyl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
2-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(dimethylamino)ethyl]-1-(2-methoxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
4-[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]-2-methoxypyridine-3-carbonitrile
methyl 6-(3-chlorobenzoyl)-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{5-[2-(4-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}-3-(1,2-oxazinan-2-yl)propanamide
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-methoxypropan-1-one
2-[(2-chlorophenyl)methyl]-N-(prop-2-en-1-yl)morpholine-4-carboxamide
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-6-methylpyridazin-3-amine
5-(3-fluorophenyl)-4-[1-(1H-imidazole-4-carbonyl)piperidin-4-yl]-2-[(2-methoxyethyl)sulfanyl]pyrimidine
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-3-(1-methylpiperidin-3-yl)propanamide
(3S)-1-{5-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1-methyl-1H-1,3-benzodiazol-2-yl}pyrrolidin-3-ol
N-[(2S)-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-oxopropan-2-yl]acetamide
[2-({4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
N-(1-methoxypropan-2-yl)-3-{[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}benzamide
6-[1-(3-chloropyridin-2-yl)piperidin-3-yl]-2-methylpyrimidin-4-ol
2-[4-(2,4-dimethoxypyrimidin-5-yl)-1H-pyrazol-1-yl]-N-(1-ethyl-1H-1,2,3-triazol-4-yl)acetamide
5-cyclobutanecarbonyl-1'-(2-methylfuran-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-methoxy-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[2-(oxolan-2-ylmethoxy)phenyl]-3-[(2,4,5-trifluorophenyl)methyl]urea
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
6-{[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3,4-dimethoxyphenyl)methyl]-N,3,5-trimethyl-1-benzofuran-2-carboxamide
2-(3-fluorophenyl)-N-({7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
N-cyclopropyl-3-[5-(3-phenylbutyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
(2S,4R)-4-(4-{[1-(2-chloro-5-fluorophenyl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(5-fluoropyridin-2-yl)pyrrolidin-3-yl]methanol
N,6-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine