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1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-1-propylpyrrolidin-2-one
(2S)-1-{5-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}propan-2-ol
5-{2-[2-(dimethylamino)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}-1-methyl-1H-pyrrole-3-carbonitrile
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[3-(3-methylphenoxy)azetidin-1-yl]ethan-1-one
3-[2-methoxy-2-(thiophen-2-yl)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-methyl-N-(2-{4-[(2-methylpyrimidin-5-yl)methyl]morpholin-2-yl}ethyl)but-2-enamide
3-hydroxy-3-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-methylpentane-1,2-dione
N-[4-(3-methoxyphenyl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
8-[1-(thiophene-2-carbonyl)piperidin-4-yl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
4-(2-methoxypyridin-3-yl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
4-(benzyloxy)-1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)piperidine
4-{5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
3-{2-[(dimethylamino)methyl]phenyl}-5-[(propan-2-yl)sulfamoyl]benzoic acid
1-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl]-4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine
8-(4-oxo-3,4-dihydrophthalazine-1-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
6-methyl-2-oxo-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-dihydroquinoline-4-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2-(2-oxopyrrolidin-1-yl)propanamide
3-[5-(4-methylphenyl)-1,3,4-thiadiazol-2-yl]-1-(piperidin-3-yl)urea
methyl[(3-methylpyridin-4-yl)methyl]{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
6-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)quinoxaline
N-[(2R)-1-hydroxy-1,1-diphenylpropan-2-yl]-2-(methylamino)pyrimidine-5-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
1-(4-{1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-4-yl}-1,4-diazepan-1-yl)ethan-1-one
(4aR,7aS)-1-cyclopropanecarbonyl-4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4S)-4-amino-N-ethyl-1-(2-hydroxy-4-methoxybenzoyl)pyrrolidine-2-carboxamide
(3S,4S)-4-propyl-1-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]pyrrolidine-3-carboxylic acid
3-(5-fluoro-2-methylphenyl)-4-methoxy-N-methylbenzamide
1-cyclohexanecarbonyl-N-[(5-methylpyrazin-2-yl)methyl]pyrrolidine-2-carboxamide
5-tert-butyl-4-{[(3S,4R)-3-methanesulfonamido-4-(propan-2-yl)pyrrolidin-1-yl]methyl}furan-2-carboxamide
(4aS,7aR)-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-fluorophenyl)-1-{5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidine
N,N-dimethyl-1-[({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)methyl]cyclohexan-1-amine
2-[(1r,4r)-4-hydroxycyclohexyl]-9-(1,3-thiazol-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-chloro-2,4-difluorophenyl)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
(3S,4R)-N,N-dimethyl-4-propyl-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-amine
4-(2,3-dihydro-1H-inden-2-yl)-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]piperazin-2-one
2-(4-chlorophenyl)-5-(2,5-dimethylfuran-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-{4-[(4-cyclopentylpiperazin-1-yl)methyl]phenyl}-2-methylbutan-2-ol
2-{[(1R,5S,6R)-3-[(2E)-hex-2-en-1-yl]-3-azabicyclo[3.1.0]hexan-6-yl]formamido}acetamide
3-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[4-(oxolan-2-ylmethoxy)phenyl]urea
(3aR,6aR)-2-cyclopropanecarbonyl-5-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-fluoro-N-{[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-3-yl]methyl}benzamide
1-[(2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-(4-methylphenyl)urea
4-[(2S)-2-hydroxypropanoyl]-1-(2-methoxyphenyl)piperazin-2-one
N-[(3R,4S)-4-cyclopropyl-1-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]pyrrolidin-3-yl]-2-ethoxyacetamide
N-[1-(3-phenylpropyl)piperidin-3-yl]cyclohex-1-ene-1-carboxamide