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N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-4-methyl-N-[(3S)-2-oxoazepan-3-yl]-1,2,5-oxadiazole-3-carboxamide
1-(2-phenoxyethyl)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2,3-dimethyl-1H-indole-7-carboxamide
1-(1H-1,2,3-benzotriazol-5-yl)-3-cyclopropyl-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}-N-[1-(thiophen-2-yl)propan-2-yl]propanamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H-indole-6-carboxamide
4-(4-ethoxy-3-methylphenyl)-N-[2-(morpholin-4-yl)ethyl]-4-oxobutanamide
methyl 6-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(2-methoxyphenyl)-2-(1-methylpyrrolidin-3-yl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]oxane-4-carboxamide
2-(6-methoxynaphthalen-2-yl)-4-(1,3-thiazol-2-ylmethyl)morpholine
5-({[(4-methyl-2-oxo-2H-chromen-7-yl)methyl](propan-2-yl)amino}methyl)pyrrolidin-2-one
N-(2-hydroxypyridin-3-yl)azocane-1-carboxamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]oxolane-3-carboxamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-4,4,4-trifluorobutanamide
(1S,6R)-9-{[5-(1,2-oxazol-5-yl)furan-2-yl]sulfonyl}-3,9-diazabicyclo[4.2.1]nonane
6-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
5-(3-acetylphenoxymethyl)-N-(cyclopropylmethyl)-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
(3aS,6aS)-2-ethyl-1-oxo-5-[3-(thiophen-3-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{5-[3-(dimethyl-1,2-oxazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridin-2-yl}acetamide
2-methoxy-6-[(4-{1-[(2-methoxyethyl)(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)methyl]phenol
(3S)-4-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-1,3-dimethylpiperazin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
N-(3-{[(2-methanesulfonylethyl)carbamoyl]amino}-4-methoxyphenyl)acetamide
1-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-{4-[3-(1H-pyrazol-1-yl)benzoyl]piperazin-1-yl}pyrimidine
5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-(1,2-oxazolidin-2-yl)pyridine
1-(4-cyclohexylpiperazin-1-yl)-2-(1H-pyrazol-1-yl)butan-1-one
1-{2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}azepan-2-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-6-(morpholin-4-yl)pyrimidin-4-amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,3,4,9-tetrahydro-1H-carbazole
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-(oxan-4-yl)-1H-1,3-benzodiazole-5-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-propylbenzamide
N'-benzyl-N-(4-fluorophenyl)-N'-(3-hydroxy-2-methylpropyl)ethanediamide
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]oxolane-2-carboxamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
3-(piperidine-1-sulfonyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide
(1S,5R)-6-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1,4-dioxan-2-ylmethyl)-N-methyl-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-(5-fluoro-1H-indol-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-({methyl[(3-phenyl-1H-pyrazol-5-yl)methyl]amino}methyl)pyridine-3-carboxylic acid
ethyl 5-{[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
4-[(2-ethylpyrimidin-4-yl)methyl]-3-(4-fluorophenyl)piperazin-2-one
methyl 3-{[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]amino}propanoate
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[2-(trifluoromethyl)morpholine-4-carbonyl]benzonitrile
4-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one