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N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
4-(3,5-dichlorobenzoyl)-1-(4-methoxyphenyl)piperazin-2-one
3-[2-(azocan-1-yl)-2-oxoethyl]-4-cyclopentylpiperazin-2-one
N-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)methyl]-2-(5,6,7,8-tetrahydronaphthalen-2-yloxy)butanamide
7-fluoro-2-methyl-3-{[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole
N-(2-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
4-{1-[(2,2-diphenylcyclopropyl)methyl]azetidin-3-yl}pyridine
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(1H-pyrazol-1-yl)butanamide
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-2,6,8-trimethylquinoline
5-(2,4-dimethoxyphenyl)-3-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-1,2,4-triazine
4-hydroxy-1-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)piperidine-4-carboxylic acid
3-cyclopentyl-1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
5-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}phenyl)-1H-pyrazole
methyl 2-(1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-oxopiperazin-2-yl)acetate
ethyl 3-(3-phenylpropyl)-1-[3-(1H-pyrazol-1-yl)propanoyl]piperidine-3-carboxylate
6-(3-methanesulfonylbenzoyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-ethyl-4-({2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}methyl)piperazin-2-one
N-{2-[5-(3-chloro-5-fluorophenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
1-(2,3,4-trifluorobenzoyl)-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
2-(morpholin-3-yl)-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)acetamide
2-[4-(5-chloropyridin-2-yl)piperazine-1-carbonyl]-3-ethyl-1H-indole
1'-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{[4-(2,6-dimethoxyphenyl)phenyl]methyl}piperidine
N-(2-fluoroethyl)-3-{[1-(6-methylpyridin-3-yl)ethyl]sulfamoyl}benzamide
N-methyl-2-[4-(pyrimidin-2-yl)piperazin-1-yl]-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
[2-methyl-2-(morpholin-4-yl)propyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(4aS,7aR)-1-(3-hydroxybenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[7-(4-methyl-1H-imidazole-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-3-ol
5-(4,6-dimethoxypyrimidin-2-yl)isoquinoline
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane
N-cyclopropyl-1-[1-(3-hydroxypyridine-2-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-(cyclohex-3-en-1-ylmethyl)-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
1-cyclopentanecarbonyl-N-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-amine
3-{6-amino-5-cyano-4-[4-(4-hydroxybut-1-yn-1-yl)phenyl]pyridin-2-yl}-1H-pyrazole-5-carboxylic acid
N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]furan-3-carboxamide
N-[3-(2-fluorophenyl)propyl]pyrimidin-2-amine
5-[3-(1-methyl-1H-pyrazol-5-yl)phenyl]pyrazine-2-carboxylic acid
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-1-(4-methoxyphenyl)cyclopentane-1-carboxamide
N-{1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl]({[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl})(pyridin-3-ylmethyl)amine
N-[2-(2-phenoxyethoxy)phenyl]oxane-4-carboxamide
(3aR,5S,6S,7aS)-2-(2-methyl-4-phenylpyrimidine-5-carbonyl)-octahydro-1H-isoindole-5,6-diol
5-fluoro-3-methyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
3-(1-cyclopropanecarbonylpiperidin-3-yl)-N-[(2,4-dimethoxyphenyl)methyl]propanamide
N-(isoquinolin-5-ylmethyl)-2,6-dimethoxy-N-methylpyridine-3-carboxamide
5-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
(1S,5R)-3-[2-(2-methylphenyl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-[2-(pyrazin-2-yl)ethyl]pyrrolidine-3-carboxamide