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1-(4-chloro-1H-pyrazole-3-carbonyl)-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
[4-({4-[3-(furan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)phenyl]methanol
3-(3-methoxyphenyl)-N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-1H-pyrazole-4-carboxamide
1-(3-fluorophenyl)-3-{1-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-methyl-4-{5-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}piperidine
N-(1,3-benzothiazol-2-ylmethyl)-6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-3-(3-methylbut-2-en-1-yl)piperidin-3-yl}methanol
1-[(3-methoxyphenyl)methyl]-4-(2-methylpropyl)-1,4-diazepan-5-one
2-(dimethylamino)-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-(4-methylphenyl)acetamide
7-{2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-[4-(pyrrolidin-1-ylmethyl)phenyl]-1H-imidazole
N-[3-(4-methoxyphenyl)propyl]-5-methyl-1,3,4-oxadiazol-2-amine
N-(2H-1,3-benzodioxol-5-yl)-3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carboxamide
2-(2,4-dimethoxyphenyl)-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]acetic acid
2-(5-acetylthiophen-3-yl)-N-cyclopentyl-N-[(2-methoxyphenyl)methyl]acetamide
2-methoxy-4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carbonitrile
N-[(2,3-dimethoxyphenyl)methyl]-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-methyl-4-(piperidin-1-ylmethyl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)benzamide
6-methyl-2-(1-methyl-1H-pyrazol-4-yl)-4-[2-(pyridin-3-ylmethyl)pyrrolidine-1-carbonyl]quinoline
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-cyclopropyl-3-({2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}sulfamoyl)benzamide
N-methyl-3-(piperidin-3-yl)-N-(quinoxalin-2-ylmethyl)benzamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(2-methylphenyl)propan-1-one
4-(4-chloro-2-methylbenzoyl)-1-(4-methylphenyl)piperazin-2-one
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-hydroxyethan-1-one
(1-benzofuran-2-ylmethyl)(methyl)[(3-methylpyridin-4-yl)methyl]amine
2-(2H-1,3-benzodioxol-5-yl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
4-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-4-oxobutane-1-sulfonamide
3-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-3-(4-methoxyphenyl)-1-(3-methylbutyl)pyrrolidine-2,5-dione
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
(1R,5R)-6-(1-benzofuran-2-ylmethyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-benzyl-3-methyl-8-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-phenyl-5-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]pentane-1,5-dione
1-ethyl-8-[(3-hydroxyphenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[4-(propan-2-yl)phenyl]urea
2-amino-6-cyclopropyl-4-(1-ethyl-5-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
7-(cyclopropylmethyl)-2-(2-methoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
2-amino-6-(2,2-dimethyloxan-4-yl)-4-[2-(ethylamino)pyrimidin-5-yl]-5-propylpyridine-3-carbonitrile
methyl 3-{[4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]amino}benzoate
1-(furan-2-yl)-2-(3-{3-[methyl(2-methylpropyl)amino]propyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)ethane-1,2-dione
2-[3-(propan-2-yl)-5-({[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}methyl)-1H-1,2,4-triazol-1-yl]pyridine
methyl[2-(methylsulfanyl)ethyl][(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
1-benzoyl-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(3,4-difluorophenyl)-5-(2-methyloxolan-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
8-(3,4-difluorobenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(2S,4R)-1-(2,6-dimethylquinoline-3-carbonyl)-4-hydroxypyrrolidine-2-carboxylic acid
2-{5-[(4-fluorophenyl)(piperidin-1-yl)methyl]-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl}acetic acid
(4aR,8aS)-6-(oxane-4-carbonyl)-1-[(3,4,5-trifluorophenyl)methyl]-decahydro-1,6-naphthyridine
N-{1-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylpyridine-2-carboxamide