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(1S,5R)-3-(1-benzoxepine-4-carbonyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{5-[(3,5-dimethylphenyl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
N-[2-(furan-2-yl)ethyl]-1-[6-(piperidine-1-carbonyl)pyrazin-2-yl]piperidin-4-amine
1-[(1S,5R)-6-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-{[4-methoxy-3-(pyridin-3-yl)phenyl]methyl}cyclopentanamine
2-(dimethylamino)-2-(3-fluorophenyl)-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]acetamide
1-{4-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]phenyl}pyrrolidin-2-one
3-(4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)-1,2-dihydropyrazin-2-one
3-(5-methylfuran-2-yl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1H-pyrazole-5-carboxamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylmethanesulfonamide
[(3R,4R)-1-(3,4-dimethylbenzoyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
8-({4-amino-6-[(3-methylphenyl)amino]-1,3,5-triazin-2-yl}methyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-(2-{1-[2-(phenylsulfanyl)ethyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
1-{4-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
(3R,4S)-4-[ethyl({[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl})amino]oxolan-3-ol
6-cyclopropyl-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]pyrimidin-4-amine
7-(3-methoxypropanamido)-N-[2-(methylsulfanyl)phenyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
7-(5-ethoxy-2-methyl-1-benzofuran-3-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(4-methylpent-3-en-1-yl)piperidine
N-methyl-5-(naphthalen-1-yl)furan-2-carboxamide
2-(4-ethylpiperazin-1-yl)-1-[3-(phenylamino)piperidin-1-yl]ethan-1-one
N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)-2-(1H-pyrazol-1-yl)butanamide
(1R,7S)-3-(3,4-dimethylphenyl)-N-methyl-N-[(2-methylpyridin-4-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-(2,2-difluoroethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-methyl-7-{[(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}-2H-chromen-2-one
3-{2-[2-(4-chloro-1-methyl-1H-indazol-3-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-fluoro-N4,N4-dimethyl-N2-[2-(2-methyl-1H-indol-3-yl)ethyl]pyrimidine-2,4-diamine
2-(3-fluorophenyl)-N-(pyridin-4-ylmethyl)-1,3-benzoxazole-5-carboxamide
4-(5-chloro-2-methoxyphenyl)-3-(1-methylpiperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,4R)-1-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-(4-acetylphenyl)-3-(4-phenylbenzoyl)piperidine-1-carboxamide
4,6-dimethyl-2-oxo-N-[2-(4,5,6,7-tetrahydro-1H-indazol-3-yl)ethyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N,N,5-trimethyl-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-methyl-1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-ol
6-cyclopentyl-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
({5-[1-(4-fluorophenyl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methyl)dimethylamine
1-(3-fluorophenyl)-N-[(3-fluorophenyl)methyl]-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-(1H-imidazol-2-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)phenyl]-5-ethyl-6-methyl-3,4-dihydropyrimidin-4-one
3-methyl-3-phenyl-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}butanamide
(2S)-1-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}pyrrolidine-2-carboxamide
2-[3-(4-methoxyphenyl)-1-(3-methylbutyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(quinoxalin-6-ylmethyl)acetamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(pyridin-4-yl)ethyl]benzamide
N-{5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,3-thiazol-2-yl}acetamide
4-(2-methylpropyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-chloro-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
(2R,6R)-4-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
methyl 5-{[(3-chlorophenyl)methyl]amino}-1-(2-methoxyethyl)-3-(3-methylbutanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-cyclopropyl-5-[4-(1-hydroxy-2-phenylethyl)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
3-(4-hydroxyphenyl)-5-[(propan-2-yl)sulfamoyl]benzoic acid