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1-({3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}methyl)azepane
(4aR,7aS)-1-benzyl-4-(5-methyl-1,3-oxazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(4-methylpiperazine-1-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(4-methyl-1H-imidazol-5-yl)methyl]-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
2-methyl-5-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
4,6-dimethyl-5-{4-[(4-methylphenyl)methyl]-3-oxopiperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidin-2-one
2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-6-methylpyridine-3-carboxylic acid
(3R,4S)-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1H-pyrazol-1-yl)butan-1-one
(4S,4aS,8aS)-4-phenyl-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-decahydroquinolin-4-ol
6-(2,3-dihydro-1,4-benzodioxin-6-yl)quinazolin-4-amine
3-({[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl)amino}methyl)benzoic acid
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-[(1R,5S,8R)-8-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]-2-(3-hydroxyphenyl)ethan-1-one
1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-N-[3-(3-methoxyphenyl)phenyl]piperidine-2-carboxamide
(3S,4S)-1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4-(1,4-oxazepan-4-yl)pyrrolidin-3-ol
5-{imidazo[1,2-a]pyrimidin-2-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methylpropanamide
4-{3-[2-(dimethylamino)ethyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-4-oxobutane-1-sulfonamide
4-{[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]methyl}-1-(propan-2-yl)pyrrolidin-2-one
4-(1-methyl-1H-pyrazol-4-yl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}pyrimidin-2-amine
3-{[(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)oxy]methyl}pyridine
4-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}pyridine
1-[(4-fluorophenyl)methyl]-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(methylsulfanyl)propan-1-one
N-{[1-(oxane-4-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
(3R,4S)-1-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-3,4-dimethylpiperidin-4-ol
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]propanamide
2-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]phenol
2-({2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}methyl)-3,5-dimethyl-1,4-dihydropyridin-4-one
N-[2-methoxy-4-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamido)phenyl]-3-methylbutanamide
N-tert-butyl-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
4-({3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzamide
N-[(5-ethylpyridin-2-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}piperidin-2-one
1-(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-2-phenoxyethan-1-one
2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-2-(1H-1,2,4-triazol-3-yl)benzamide
N-cyclopropyl-5-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-ethyl-4-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}pyrimidine
2-(1H-indol-4-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[5-(diphenylmethyl)-1,2,4-oxadiazol-3-yl]pyridazine
7-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
3-methoxy-1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperidine
3-(3-methoxypropyl)-1-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetyl]piperidine-3-carboxylic acid
[3-(2H-1,3-benzodioxol-5-yl)propyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
5-(6-methylpyridazin-3-yl)-1,2,3,4-tetrahydroisoquinoline