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2-(4-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one
2-{3-[(3-chlorophenyl)methyl]-5-[(pyridin-4-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
[(3R,4R)-4-[({[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}amino)methyl]pyrrolidin-3-yl]methanol
1-[3-(4-fluorophenoxy)azetidine-1-carbonyl]cyclopropane-1-carboxamide
1-(1-cyclopentylpiperidin-3-yl)-4-(2-methylphenyl)piperazine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl 5-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-3-cyclobutaneamido-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(3-phenoxyphenyl)-4H-1,2,4-triazole
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(4-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-methyl-N-[2-(5-methylfuran-2-yl)ethyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
6-ethyl-N,1,5-trimethyl-2-oxo-N-[1-(pyridin-2-yl)propyl]-1,2-dihydropyridine-3-carboxamide
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-(3-methylbut-2-en-1-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-cyclooctyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-1,3-thiazole-4-carboxamide
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1H-imidazole-2-carboxamide
butyl 4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carboxylate
N-{4-chloro-3-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]phenyl}acetamide
N-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
{4-[(2-chlorophenyl)methyl]-1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl}methanol
ethyl N-[(3S,5S)-5-{[(3-chlorophenyl)methyl]carbamoyl}-1-methylpyrrolidin-3-yl]carbamate
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[(3-propylmorpholin-4-yl)methyl]benzoic acid
1-(1-benzofuran-2-ylmethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
(3aR,6aR)-2-acetyl-5-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-chlorophenyl)-3-{[1-(2-methoxyacetyl)piperidin-4-yl]formamido}propanoic acid
2-(4-fluorophenyl)-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)acetamide
{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
N-cyclopentyl-N'-[(2,4-dimethoxyphenyl)methyl]butanediamide
1-{4-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-(4-methoxyphenyl)-1H-pyrazole
1-methyl-6-propyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[2-(pyrazin-2-yl)ethyl]piperidine-3-carboxamide
N-{1-[7-acetyl-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperidin-4-yl}acetamide
1-methyl-3-[3-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxymethyl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
1-(2,3-difluoro-6-methoxybenzoyl)-4-(piperidine-1-carbonyl)piperidine
N-(2,5-dimethylphenyl)-2-(1H-imidazol-4-ylmethyl)-3-oxopiperazine-1-carboxamide
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(1H-imidazol-2-yl)piperidine
4-(2,4-dioxoimidazolidin-1-yl)-N-({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)benzamide
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}propanamide
(2S,4R)-4-amino-N-methyl-1-({4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}methyl)pyrrolidine-2-carboxamide
2-(cyclopropylmethyl)-7-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-{3-[1-(2-phenoxyethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
2-[2-(1H-imidazol-4-yl)ethyl]-9-(4,4,4-trifluorobutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-4-amine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
4-[3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)propyl]piperazin-2-one
2-(3,4-dimethylphenoxy)-1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
N,6-dimethyl-2-oxo-N-(propan-2-yl)-4-[2-(propylamino)pyrimidin-5-yl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide